Guo Liangqin, Ye Zhixiong, Ujjainwalla Feroze, Sings Heather L, Sebhat Iyassu K, Huber John, Weinberg David H, Tang Rui, MacNeil Tanya, Tamvakopoulos Constantin, Peng Qianping, MacIntyre Euan, van der Ploeg Lex H T, Goulet Mark T, Wyvratt Matthew J, Nargund Ravi P
Department of Medicinal Chemistry, Merck Research Laboratories, 126 E. Lincoln Avenue, PO Box 2000, RY 50G-332, Rahway, NJ 07065, USA.
Bioorg Med Chem Lett. 2008 Jun 1;18(11):3242-7. doi: 10.1016/j.bmcl.2008.04.049. Epub 2008 Apr 25.
Discovery of a series of tert-butyl pyrrolidine derived, potent and orally bioavailable melanocortin receptor subtype-4 (MC4R) selective modulators is disclosed.
公开了一系列源自叔丁基吡咯烷的、强效且口服生物可利用的黑皮质素受体亚型-4（MC4R）选择性调节剂的发现。
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