芳基肼基氰基丙烯酸酯和N-芳基吡唑羧酸酯的合成与生物学评价
Synthesis and biological evaluation of arylhydrazinocyanoacrylates and N-aryl pyrazolecarboxylates.
作者信息
Liu Yuxiu, Liu Shaohua, Li Yonghong, Song Haibin, Wang Qingmin
机构信息
State Key Laboratory of Elemento-Organic Chemistry, Institute of Elemento-Organic Chemistry, Nankai University, Tianjin, China.
出版信息
Bioorg Med Chem Lett. 2009 Jun 1;19(11):2953-6. doi: 10.1016/j.bmcl.2009.04.048. Epub 2009 Apr 18.
PMID:19406637
Abstract
A series of arylhydrazino-substituted cyanoacrylates 3 and N-aryl pyrazolecarboxylates 6 were synthesized and their bioactivities were evaluated. Though compounds 3 were designed as herbicide, some of them showed fungicidal activity and anti-tumor activity. Some of the compounds 6 exhibited plant growth regulatory activity.
摘要
合成了一系列芳基肼基取代的氰基丙烯酸酯3和N-芳基吡唑羧酸酯6，并对其生物活性进行了评价。虽然化合物3被设计为除草剂，但其中一些表现出杀菌活性和抗肿瘤活性。一些化合物6表现出植物生长调节活性。
Zotero 插件