Yoshida K, Horikoshi Y, Eta M, Chikazawa J, Ogishima M, Fukuda Y, Sato H
Central Research Laboratories, Zeria Pharmaceutical Co., Ltd., Saitama, Japan.
Bioorg Med Chem Lett. 1998 Nov 3;8(21):2967-72. doi: 10.1016/S0960-894X(98)00538-1.
Synthesis of benzanilide derivatives which have dual alpha 1-adrenoceptor antagonistic action and steroid 5 alpha-reductase inhibitory activity and their structure-activity relationships is described.