脂肪细胞中β-肾上腺素能受体拮抗剂与受体相互作用的立体化学方面。人和大鼠脂肪细胞中β-肾上腺素能受体的分化。 - Suppr

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超能文献

Stereochemical aspects of beta-adrenoceptor antagonist-receptor interaction in adipocytes. Differentiation of beta-adrenoceptors in human and rat adipocytes.

作者信息

Harms H H

出版信息

Life Sci. 1976 Nov 1;19(9):1447-52. doi: 10.1016/0024-3205(76)90447-1.

DOI:10.1016/0024-3205(76)90447-1

PMID:11387

Abstract

摘要

相似文献

Stereochemical aspects of beta-adrenoceptor antagonist-receptor interaction in adipocytes. Differentiation of beta-adrenoceptors in human and rat adipocytes.脂肪细胞中β-肾上腺素能受体拮抗剂与受体相互作用的立体化学方面。人和大鼠脂肪细胞中β-肾上腺素能受体的分化。

Life Sci. 1976 Nov 1;19(9):1447-52. doi: 10.1016/0024-3205(76)90447-1.

Differentiation of beta-adrenoceptors in right atrium, diaphragm and adipose tissue of the rat, using stereoisomers of propranolol, alprenolol, nifenalol and practolol.使用普萘洛尔、阿普洛尔、硝苯洛尔和醋丁洛尔的立体异构体对大鼠右心房、膈肌和脂肪组织中的β-肾上腺素能受体进行鉴别。

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Species and strain-related differences in the expression and functionality of beta-adrenoceptor subtypes in adipose tissue.脂肪组织中β-肾上腺素能受体亚型表达及功能的物种和品系相关差异。

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The effects of beta-adrenoceptor blocking drugs on non-esterified fatty acid release from adipocytes.β-肾上腺素能受体阻断药物对脂肪细胞非酯化脂肪酸释放的影响。

J Pharmacol. 1983;14 Suppl 2:209-15.

Evaluation of beta adrenoceptor antagonist affinity and cardioselectivity by radioligand-receptor assay.通过放射性配体-受体分析法评估β肾上腺素能受体拮抗剂的亲和力和心脏选择性。

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Coexistence of beta1 and beta2 adrenoceptors in mammalian lung: evidence from direct binding studies.哺乳动物肺中β1和β2肾上腺素能受体的共存：直接结合研究的证据。

Mol Pharmacol. 1978 Nov;14(6):996-1005.

Comparison of specificity of agonist and antagonist radioligand binding to beta adrenergic receptors.激动剂和拮抗剂放射性配体与β肾上腺素能受体结合特异性的比较。

Nature. 1977 Aug 4;268(5619):453-4. doi: 10.1038/268453a0.

Disposition and activity of beta-adrenoceptor antagonists in the rat using an ex vivo receptor binding assay.使用体外受体结合试验研究大鼠体内β-肾上腺素能受体拮抗剂的分布与活性。

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Identity of [3H]dihydroalprenolol binding sites and beta-2 adrenergic receptors coupled with adenylate cyclase in guinea-pig skeletal muscle sarcolemma: general properties and structure-activity relationships.豚鼠骨骼肌肌膜中[3H]二氢阿普洛尔结合位点及与腺苷酸环化酶偶联的β-2肾上腺素能受体的特性：一般性质及构效关系

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beta-Adrenoceptor studies. 6. Further investigations on the hybrid nature of the rat adipocyte beta-adrenoceptor.β-肾上腺素能受体研究。6. 对大鼠脂肪细胞β-肾上腺素能受体杂交性质的进一步研究。

Eur J Pharmacol. 1980 Apr 11;63(1):73-83. doi: 10.1016/0014-2999(80)90118-1.

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Atypical characteristics of the beta-adrenoceptor mediating cyclic AMP generation and lipolysis in the rat adipocyte.介导大鼠脂肪细胞中环磷酸腺苷生成及脂肪分解的β-肾上腺素能受体的非典型特征。

Br J Pharmacol. 1985 Jan;84(1):131-7.

Blockade of isoprenaline-induced changes in plasma free fatty acids, immunoreactive insulin levels and plasma renin activity in healthy human subjects, by propranolol, pindolol, practolol, atenolol, metoprolol and acebutolol.普萘洛尔、吲哚洛尔、醋氨心安、阿替洛尔、美托洛尔和醋丁洛尔对健康人体受试者中异丙肾上腺素诱导的血浆游离脂肪酸、免疫反应性胰岛素水平和血浆肾素活性变化的阻断作用。

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