Fernández-Gacio Ana, Fernández-Marcos Carlos, Swamy Narasimha, Ray Rahul
Bioorganic Chemistry and Structural Biology, Section in Endocrinology, Diabetes and Metabolism, Department of Medicine, Boston University School of Medicine, 85 East Newton Street, Boston, MA 02118, USA.
Bioorg Med Chem Lett. 2003 Jan 20;13(2):213-6. doi: 10.1016/s0960-894x(02)00878-8.
Synthesis of an affinity alkylating non steroidal mimic of 1alpha,25-dihydroxyvitamin D(3) and its radiolabeled counterpart is presented. We also report the affinity labeling of the VDR-ligand binding domain (VDR-LBD) with this analogue.
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