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A mimicry of primary amines by bis-secondary diamines as components in the Ugi four-component reaction.

作者信息

Giovenzana Giovanni Battista, Tron Gian Cesare, Di Paola Stefano, Menegotto Ivan Guglielmo, Pirali Tracey

机构信息

Di.S.C.A.F.F. and Drug and Food Biotechnology Center, Università degli Studi del Piemonte Orientale A. Avogadro, Via Bovio 6, 28100 Novara, Italy.

出版信息

Angew Chem Int Ed Engl. 2006 Feb 6;45(7):1099-102. doi: 10.1002/anie.200503095.

DOI:10.1002/anie.200503095

PMID:16389629

Abstract

摘要

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A mimicry of primary amines by bis-secondary diamines as components in the Ugi four-component reaction.

作者信息

Giovenzana Giovanni Battista, Tron Gian Cesare, Di Paola Stefano, Menegotto Ivan Guglielmo, Pirali Tracey

机构信息

Di.S.C.A.F.F. and Drug and Food Biotechnology Center, Università degli Studi del Piemonte Orientale A. Avogadro, Via Bovio 6, 28100 Novara, Italy.

出版信息

Angew Chem Int Ed Engl. 2006 Feb 6;45(7):1099-102. doi: 10.1002/anie.200503095.

DOI:10.1002/anie.200503095

PMID:16389629

Abstract

摘要

相似文献

A mimicry of primary amines by bis-secondary diamines as components in the Ugi four-component reaction.

Angew Chem Int Ed Engl. 2006 Feb 6;45(7):1099-102. doi: 10.1002/anie.200503095.

The use of the Ugi four-component condensation.

Nat Protoc. 2007;2(3):632-9. doi: 10.1038/nprot.2007.71.

Brønsted acid-catalyzed efficient Strecker reaction of ketones, amines and trimethylsilyl cyanide.

Org Biomol Chem. 2010 Mar 21;8(6):1399-405. doi: 10.1039/b924272d. Epub 2010 Jan 20.

Catalytic asymmetric three-component acyl-Strecker reaction.

Org Lett. 2007 Mar 15;9(6):1149-51. doi: 10.1021/ol0702674. Epub 2007 Feb 24.

Synthesis of (S)- and (R)-5-oxo-piperazine-2-carboxylic acid and its application to peptidomimetics.

J Org Chem. 2009 Nov 6;74(21):8433-6. doi: 10.1021/jo901389q.

Probing the mechanism of the Ugi four-component reaction with charge-tagged reagents by ESI-MS(/MS).

Chem Commun (Camb). 2014 Jan 11;50(3):338-40. doi: 10.1039/c3cc47156j. Epub 2013 Nov 15.

Determination of the enantiomeric excess of chiral carboxylic acids by 31P NMR with phosphorylated derivatizing agents from C2-symmetrical diamines containing the (S)-alpha-phenylethyl group.

Chirality. 2007 Jun;19(6):503-7. doi: 10.1002/chir.20406.

Diversity oriented and chemoenzymatic synthesis of densely functionalized pyrrolidines through a highly diastereoselective Ugi multicomponent reaction.

Org Biomol Chem. 2012 Feb 14;10(6):1255-74. doi: 10.1039/c1ob06632c. Epub 2012 Jan 4.

The catalytic acylcyanation of imines.

Chem Asian J. 2008 Feb 1;3(2):430-7. doi: 10.1002/asia.200700327.

An efficient synthesis of symmetric and unsymmetric bis-(β-aminoamides) via Ugi multicomponent reaction.

Org Lett. 2012 Dec 7;14(23):6044-7. doi: 10.1021/ol302935y. Epub 2012 Nov 14.

引用本文的文献

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Nat Commun. 2025 Apr 29;16(1):4021. doi: 10.1038/s41467-025-59136-z.

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FEBS J. 2025 Jul;292(13):3449-3476. doi: 10.1111/febs.70065. Epub 2025 Mar 23.

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Org Lett. 2025 Feb 28;27(8):1829-1834. doi: 10.1021/acs.orglett.4c04810. Epub 2025 Feb 17.

Versatile One-Pot Synthesis of Hydrophobic Tags by Multicomponent Reactions.

ACS Omega. 2025 Jan 30;10(5):4745-4753. doi: 10.1021/acsomega.4c09726. eCollection 2025 Feb 11.

Harnessing unprotected deactivated amines and arylglyoxals in the Ugi reaction for the synthesis of fused complex nitrogen heterocycles.

Beilstein J Org Chem. 2024 Jul 25;20:1758-1766. doi: 10.3762/bjoc.20.154. eCollection 2024.

A Versatile and Sustainable Multicomponent Platform for the Synthesis of Protein Degraders: Proof-of-Concept Application to BRD4-Degrading PROTACs.

J Med Chem. 2022 Nov 2;65(22):15282-99. doi: 10.1021/acs.jmedchem.2c01218.

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Molecules. 2022 Sep 21;27(19):6218. doi: 10.3390/molecules27196218.

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Molecules. 2021 Oct 30;26(21):6579. doi: 10.3390/molecules26216579.

Multicomponent reaction-derived covalent inhibitor space.

Sci Adv. 2021 Feb 3;7(6). doi: 10.1126/sciadv.abd9307. Print 2021 Feb.

A One-Pot Synthesis of Oxazepine-Quinazolinone bis-Heterocyclic Scaffolds via Isocyanide-Based Three-Component Reactions.

Front Chem. 2019 Sep 18;7:623. doi: 10.3389/fchem.2019.00623. eCollection 2019.

A mimicry of primary amines by bis-secondary diamines as components in the Ugi four-component reaction.

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A mimicry of primary amines by bis-secondary diamines as components in the Ugi four-component reaction.

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出版信息

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