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Discovery of 1-(2,4-dichlorophenyl)-4-ethyl-5-(5-(2-(4-(trifluoromethyl)phenyl)ethynyl)thiophen-2-yl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide as a potential peripheral cannabinoid-1 receptor inverse agonist.

作者信息

Hung Ming-Shiu, Chang Chun-Ping, Li Ting-Chieh, Yeh Teng-Kuang, Song Jen-Shin, Lin Yinchiu, Wu Chien-Huang, Kuo Po-Chu, Amancha Prashanth K, Wong Ying-Chieh, Hsiao Wen-Chi, Chao Yu-Sheng, Shia Kak-Shan

机构信息

Division of Biotechnology and Pharmaceutical Research, National Health Research Institutes, 35, Keyan Road, Zhunan Town, Miaoli County 35053, Taiwan, ROC.

出版信息

ChemMedChem. 2010 Sep 3;5(9):1439-43. doi: 10.1002/cmdc.201000246.

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