Institute of Life Sciences, University of Hyderabad Campus, Gachibowli, Hyderabad 500 046, India.
Chem Commun (Camb). 2013 Jan 7;49(2):190-2. doi: 10.1039/c2cc37070k. Epub 2012 Nov 21.
A rapid, versatile and one-pot Cu-mediated domino reaction has been developed for facile assembly of two six membered fused N-heterocyclic rings leading to novel small molecules as potential inhibitors of PDE4.
一种快速、多功能且一锅法的 Cu 介导的级联反应已经被开发出来,用于简便地组装两个六元融合的 N-杂环,得到新型小分子,作为潜在的 PDE4 抑制剂。