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Experience with ponatinib in paediatric patients with leukaemia.
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Ponatinib (AP24534) is a novel potent inhibitor of oncogenic RET mutants associated with thyroid cancer.
J Clin Endocrinol Metab. 2013 May;98(5):E811-9. doi: 10.1210/jc.2012-2672. Epub 2013 Mar 22.

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Decoding tumor angiogenesis: pathways, mechanisms, and future directions in anti-cancer strategies.
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Overcoming Secondary Mutations of Type II Kinase Inhibitors.
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Targeting casein kinase 1 for cancer therapy: current strategies and future perspectives.
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Vemurafenib inhibits necroptosis in normal and pathological conditions as a RIPK1 antagonist.
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Improving drug discovery with a hybrid deep generative model using reinforcement learning trained on a Bayesian docking approximation.
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Angiogenic signaling pathways and anti-angiogenic therapy for cancer.
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A phase 2 trial of ponatinib in Philadelphia chromosome-positive leukemias.
N Engl J Med. 2013 Nov 7;369(19):1783-96. doi: 10.1056/NEJMoa1306494. Epub 2013 Nov 1.
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Ponatinib in refractory Philadelphia chromosome-positive leukemias.
N Engl J Med. 2012 Nov 29;367(22):2075-88. doi: 10.1056/NEJMoa1205127.
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Accelerated approval of oncology products: the food and drug administration experience.
J Natl Cancer Inst. 2011 Apr 20;103(8):636-44. doi: 10.1093/jnci/djr062. Epub 2011 Mar 21.
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Therapeutic options against BCR-ABL1 T315I-positive chronic myelogenous leukemia.
Clin Cancer Res. 2008 Jul 15;14(14):4392-9. doi: 10.1158/1078-0432.CCR-08-0117.

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