2-Oxooxazolidine-5-carboxamides as Na1.8 Inhibitors for Treating Pain Disorders, Cough Disorders, and Acute and Chronic Itch Disorders.
作者信息
Sabnis Ram W
机构信息
Smith, Gambrell & Russell LLP, 1105 W. Peachtree Street NE, Suite 1000, Atlanta, Georgia 30309, United States.
出版信息
ACS Med Chem Lett. 2022 Mar 1;13(3):334-335. doi: 10.1021/acsmedchemlett.2c00058. eCollection 2022 Mar 10.
Abstract
摘要
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本文引用的文献
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Epigenetic Mechanisms of Neural Plasticity in Chronic Neuropathic Pain.慢性神经性疼痛中的神经可塑性的表观遗传机制。
ACS Chem Neurosci. 2022 Feb 16;13(4):432-441. doi: 10.1021/acschemneuro.1c00841. Epub 2022 Feb 2.
2
Ventricular voltage-gated ion channels: Detection, characteristics, mechanisms, and drug safety evaluation.心室电压门控离子通道：检测、特征、机制和药物安全性评价。
Clin Transl Med. 2021 Oct;11(10):e530. doi: 10.1002/ctm2.530.
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Painful diabetic peripheral neuropathy: Role of oxidative stress and central sensitisation.痛性糖尿病周围神经病：氧化应激和中枢敏化的作用。
Diabet Med. 2022 Jan;39(1):e14729. doi: 10.1111/dme.14729. Epub 2021 Oct 28.
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Novel Approaches, Drug Candidates, and Targets in Pain Drug Discovery.新型方法、候选药物和疼痛药物发现中的靶点。
J Med Chem. 2021 May 27;64(10):6523-6548. doi: 10.1021/acs.jmedchem.1c00028. Epub 2021 May 6.
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Pain behavior in SCN9A (Nav1.7) and SCN10A (Nav1.8) mutant rodent models.SCN9A（Nav1.7）和 SCN10A（Nav1.8）突变啮齿动物模型的疼痛行为。
Neurosci Lett. 2021 May 14;753:135844. doi: 10.1016/j.neulet.2021.135844. Epub 2021 Mar 26.
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Mini-review - Sodium channels and beyond in peripheral nerve disease: Modulation by cytokines and their effector protein kinases.综述 - 周围神经疾病中的钠离子通道及其他：细胞因子及其效应蛋白激酶的调节作用。
Neurosci Lett. 2021 Jan 10;741:135446. doi: 10.1016/j.neulet.2020.135446. Epub 2020 Nov 6.
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