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Novel Quinoline Compounds as EZH2 Inhibitors for Treating Cancer.

作者信息

Sabnis Ram W

机构信息

Smith, Gambrell & Russell LLP, 1105 West Peachtree Street NE, Suite 1000, Atlanta, Georgia 30309, United States.

出版信息

ACS Med Chem Lett. 2022 Apr 13;13(5):755-756. doi: 10.1021/acsmedchemlett.2c00139. eCollection 2022 May 12.

Abstract
摘要

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本文引用的文献

1
EZH2, a prominent orchestrator of genetic and epigenetic regulation of solid tumor microenvironment and immunotherapy.
Biochim Biophys Acta Rev Cancer. 2022 Mar;1877(2):188700. doi: 10.1016/j.bbcan.2022.188700. Epub 2022 Feb 22.
2
New insights into the interplay between long non-coding RNAs and RNA-binding proteins in cancer.
Cancer Commun (Lond). 2022 Feb;42(2):117-140. doi: 10.1002/cac2.12254. Epub 2022 Jan 12.
3
Non-coding RNAs-EZH2 regulatory mechanisms in cervical cancer: The current state of knowledge.
Biomed Pharmacother. 2022 Feb;146:112123. doi: 10.1016/j.biopha.2021.112123. Epub 2021 Dec 13.
4
Role of EZH2 in bone marrow mesenchymal stem cells and immune-cancer interactions.
Crit Rev Oncol Hematol. 2022 Jan;169:103547. doi: 10.1016/j.critrevonc.2021.103547. Epub 2021 Nov 26.
5
Critical role of the high mobility group A proteins in hematological malignancies.
Hematol Oncol. 2022 Feb;40(1):2-10. doi: 10.1002/hon.2934. Epub 2021 Oct 12.
6
Epigenetic regulation in medulloblastoma pathogenesis revealed by genetically engineered mouse models.
Cancer Sci. 2021 Aug;112(8):2948-2957. doi: 10.1111/cas.14990. Epub 2021 Jun 17.

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