2-（2-苯基环丙基）咪唑啉：在I(1)和I(2)咪唑啉受体处的对映选择性相互作用逆转 - Suppr

2-(2-Phenylcyclopropyl)imidazolines: reversed enantioselective interaction at I(1) and I(2) imidazoline receptors.

作者信息

Quaglia W, Bousquet P, Pigini M, Carotti A, Carrieri A, Dontenwill M, Gentili F, Giannella M, Maranca F, Piergentili A, Brasili L

机构信息

Dipartimento di Scienze Chimiche, Università di Camerino, Via S. Agostino 1, 62032 Camerino, Italy.

出版信息

J Med Chem. 1999 Jul 29;42(15):2737-40. doi: 10.1021/jm991049m.

DOI:10.1021/jm991049m

PMID:10425083

Abstract

摘要

相似文献

2-(2-Phenylcyclopropyl)imidazolines: reversed enantioselective interaction at I(1) and I(2) imidazoline receptors.2-（2-苯基环丙基）咪唑啉：在I(1)和I(2)咪唑啉受体处的对映选择性相互作用逆转

J Med Chem. 1999 Jul 29;42(15):2737-40. doi: 10.1021/jm991049m.

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Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models.配体与I2咪唑啉受体的结合：亲脂性在定量构效关系模型中的作用。

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Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives.新型2-(4,5-二氢-1H-咪唑-2-基)-3,4-二氢-2H-1,4-苯并恶嗪衍生物的合成与生物学评价

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J Med Chem. 2002 Jan 3;45(1):32-40. doi: 10.1021/jm0110082.

High-affinity binding of beta-carbolines to imidazoline I2B receptors and MAO-A in rat tissues: norharman blocks the effect of morphine withdrawal on DOPA/noradrenaline synthesis in the brain.β-咔啉与大鼠组织中咪唑啉I2B受体和单胺氧化酶A的高亲和力结合：去甲哈尔满阻断吗啡戒断对脑中多巴/去甲肾上腺素合成的影响。

Eur J Pharmacol. 2005 Aug 22;518(2-3):234-42. doi: 10.1016/j.ejphar.2005.06.023.

Preparation, structure and affinity for imidazoline I2 receptors and alpha2-adrenoceptors of 1-[(4,5-dihydroimidazolidin-2-yl)imino]indan-2-ols.1-[(4,5-二氢咪唑烷-2-基)亚氨基]茚满-2-醇对咪唑啉I2受体和α2-肾上腺素能受体的制备、结构及亲和力

Acta Pol Pharm. 2005 Nov-Dec;62(6):497-502.

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Functional studies of specific imidazoline-2 receptor ligands.

Ann N Y Acad Sci. 1995 Jul 12;763:125-39. doi: 10.1111/j.1749-6632.1995.tb32397.x.

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2-(2-Phenylcyclopropyl)imidazolines: reversed enantioselective interaction at I(1) and I(2) imidazoline receptors.

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