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Degradation kinetics of oxycarbonyloxymethyl prodrugs of phosphonates in solution.

作者信息

Yuan L C, Dahl T C, Oliyai R

机构信息

Gilead Sciences, Foster City, California 94404, USA.

出版信息

Pharm Res. 2001 Feb;18(2):234-7. doi: 10.1023/a:1011044804823.

DOI:10.1023/a:1011044804823
PMID:11405296
Abstract
摘要

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Pharm Res. 1997 Dec;14(12):1824-9. doi: 10.1023/a:1012108719462.
2
Pharmacokinetics, safety and bioavailability of HPMPC (cidofovir) in human immunodeficiency virus-infected subjects.膦甲酸钠（西多福韦）在人类免疫缺陷病毒感染受试者中的药代动力学、安全性和生物利用度。
Antiviral Res. 1996 Mar;29(2-3):153-61. doi: 10.1016/0166-3542(95)00829-2.
3
Phosphoryloxymethyl carbamates and carbonates--novel water-soluble prodrugs for amines and hindered alcohols.
A strategy for addicting transgene-free bacteria to synthetic modified metabolites.
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Front Microbiol. 2023 Feb 10;14:1086094. doi: 10.3389/fmicb.2023.1086094. eCollection 2023.
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ACS Omega. 2020 Nov 4;5(45):29373-29381. doi: 10.1021/acsomega.0c04205. eCollection 2020 Nov 17.
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Phosphonate prodrugs: an overview and recent advances.膦酸酯前药：概述及最新进展。
Future Med Chem. 2019 Jul;11(13):1625-1643. doi: 10.4155/fmc-2018-0591.
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Pharmacokinetics of tenofovir monoester and association with intracellular tenofovir diphosphate following single-dose tenofovir disoproxil fumarate.富马酸替诺福韦二吡呋酯单酯的药代动力学及其与单次给药后细胞内替诺福韦二磷酸酯的关系。
J Antimicrob Chemother. 2019 Aug 1;74(8):2352-2359. doi: 10.1093/jac/dkz187.
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Drug Des Devel Ther. 2017 Nov 6;11:3171-3177. doi: 10.2147/DDDT.S149125. eCollection 2017.
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Molecules. 2017 Jul 14;22(7):1182. doi: 10.3390/molecules22071182.
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