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In vitro glucocorticoid resistance in childhood leukemia correlates with receptor affinity determined at 37 degrees C, but not with affinity determined at room temperature.

作者信息

Haarman E G, Kaspers G J L, Pieters R, Rottier M M A, Den Boer M L, Janka-Schaub G E, Veerman A J P

出版信息

Leukemia. 2002 Sep;16(9):1882-4. doi: 10.1038/sj.leu.2402606.

DOI:10.1038/sj.leu.2402606
PMID:12200716
Abstract
摘要

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1
In vitro glucocorticoid resistance in childhood leukemia correlates with receptor affinity determined at 37 degrees C, but not with affinity determined at room temperature.儿童白血病中的体外糖皮质激素抵抗与在37摄氏度测定的受体亲和力相关,但与在室温下测定的亲和力无关。
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A case of primary glucocorticoid resistance.一例原发性糖皮质激素抵抗病例。
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Kinetics of the in vivo expression of glucocorticoid receptor splice variants during prednisone treatment in childhood acute lymphoblastic leukaemia.儿童急性淋巴细胞白血病泼尼松治疗期间糖皮质激素受体剪接变体的体内表达动力学
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Overcoming Glucocorticoid Resistance in Acute Lymphoblastic Leukemia: Repurposed Drugs Can Improve the Protocol.克服急性淋巴细胞白血病中的糖皮质激素抵抗:重新利用的药物可改善治疗方案。
Front Oncol. 2021 Mar 11;11:617937. doi: 10.3389/fonc.2021.617937. eCollection 2021.
2
Molecular pharmacodynamics in childhood leukemia.儿童白血病中的分子药效学
Int J Hematol. 2003 Dec;78(5):402-13. doi: 10.1007/BF02983812.