外部亲核试剂浓度对O-乙酰水杨酰胺分子内O到N酰化的竞争性抑制作用。 - Suppr

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超能文献

Competitive inhibitory effect of external nucleophile concentration on intramolecular O- to N-acylation in O-acetylsalicylamide.

作者信息

Hussain A A, Jona J, Crooks P A

机构信息

University of Kentucky College of Pharmacy, Lexington, KY, 40536-0082, USA.

出版信息

AAPS PharmSciTech. 2000 Aug 19;1(3):E-TN1. doi: 10.1208/pt0103_tn1.

DOI:10.1208/pt0103_tn1

PMID:14727901

原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC2750343/

Abstract

摘要

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Competitive inhibitory effect of external nucleophile concentration on intramolecular O- to N-acylation in O-acetylsalicylamide.外部亲核试剂浓度对O-乙酰水杨酰胺分子内O到N酰化的竞争性抑制作用。

AAPS PharmSciTech. 2000 Aug 19;1(3):E-TN1. doi: 10.1208/pt0103_tn1.

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本文引用的文献

Rearrangement of O-acylsalicylamides via intramolecular O-to-N transacylation: rate enhancement by an adjacent carboxylic acid group.

J Pharm Sci. 1990 Jul;79(7):651. doi: 10.1002/jps.2600790724.

Precautionary note for use of bisulfite in pharmaceutical formulations.亚硫酸氢盐在药物制剂中使用的注意事项。

J Pharm Sci. 1977 Dec;66(12):1775-6. doi: 10.1002/jps.2600661234.

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