Dunn Derek, Husten Jean, Ator Mark A, Chatterjee Sankar
Cephalon Inc., 145 Brandywine Parkway, West Chester, PA 19380-4245, USA.
Bioorg Med Chem Lett. 2007 Jan 15;17(2):542-5. doi: 10.1016/j.bmcl.2006.10.010. Epub 2006 Oct 10.
Synthesis and activity of a series of 4-thiazol-yl substituted analogs of novel pyrrolocarbazole 1 as poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors have been disclosed.
已公开了一系列新型吡咯并咔唑1的4-噻唑基取代类似物作为聚(ADP-核糖)聚合酶-1(PARP-1)抑制剂的合成及活性。