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Reversed chloroquines based on the 3,4-dihydropyrimidin-2(1H)-one scaffold: synthesis and evaluation for antimalarial, beta-haematin inhibition, and cytotoxic activity.

作者信息

October Natasha, Watermeyer Nicholas D, Yardley Vanessa, Egan Timothy J, Ncokazi Kanyile, Chibale Kelly

机构信息

Department of Chemistry, University of Cape Town, Rondebosch, South Africa.

出版信息

ChemMedChem. 2008 Nov;3(11):1649-53. doi: 10.1002/cmdc.200800172.

DOI:10.1002/cmdc.200800172
PMID:18846586
Abstract
摘要

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