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Synthesis and pharmacology of anti-inflammatory steroidal antedrugs.

作者信息

Khan M Omar F, Lee Henry J

机构信息

College of Pharmacy, Southwestern Oklahoma State University, 100 Campus Drive, Weatherford, Oklahoma 73096, USA.

出版信息

Chem Rev. 2008 Dec;108(12):5131-45. doi: 10.1021/cr068203e.

DOI:10.1021/cr068203e
PMID:19035773
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC2650492/
Abstract
摘要

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Loteprednol etabonate: clinical potential in the management of ocular inflammation.卤替泼诺酯：在眼部炎症治疗中的临床潜力。
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In vitro anti-inflammatory activities of new steroidal antedrugs: [16alpha,17alpha-d] Isoxazoline and [16alpha,17alpha-d]-3'-hydroxy-iminoformyl isoxazoline derivatives of prednisolone and 9alpha-fluoroprednisolone.新型甾体前药的体外抗炎活性：泼尼松龙和9α-氟泼尼松龙的[16α,17α-d]异恶唑啉及[16α,17α-d]-3'-羟基-亚氨基甲酰基异恶唑啉衍生物
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