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How does Viagra protect the ischemic heart?

作者信息

Xia Yong

出版信息

Am J Physiol Heart Circ Physiol. 2009 May;296(5):H1209-10. doi: 10.1152/ajpheart.00298.2009. Epub 2009 Apr 3.

Abstract
摘要

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本文引用的文献

1
ERK phosphorylation mediates sildenafil-induced myocardial protection against ischemia-reperfusion injury in mice.
Am J Physiol Heart Circ Physiol. 2009 May;296(5):H1236-43. doi: 10.1152/ajpheart.00100.2009. Epub 2009 Mar 13.
2
Exploring pluripotency with chemical genetics.
Cell Stem Cell. 2009 Feb 6;4(2):98-100. doi: 10.1016/j.stem.2009.01.005.
3
Protein kinase G-dependent cardioprotective mechanism of phosphodiesterase-5 inhibition involves phosphorylation of ERK and GSK3beta.
J Biol Chem. 2008 Oct 24;283(43):29572-85. doi: 10.1074/jbc.M801547200. Epub 2008 Aug 21.
4
Does sildenafil cause myocardial infarction or sudden cardiac death?
Am J Cardiovasc Drugs. 2008;8(1):1-7. doi: 10.2165/00129784-200808010-00001.
5
Chronic inhibition of cyclic GMP phosphodiesterase 5A prevents and reverses cardiac hypertrophy.
Nat Med. 2005 Feb;11(2):214-22. doi: 10.1038/nm1175. Epub 2005 Jan 23.
7
Sildenafil (Viagra) induces powerful cardioprotective effect via opening of mitochondrial K(ATP) channels in rabbits.
Am J Physiol Heart Circ Physiol. 2002 Sep;283(3):H1263-9. doi: 10.1152/ajpheart.00324.2002.
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Specificity and mechanism of action of some commonly used protein kinase inhibitors.
Biochem J. 2000 Oct 1;351(Pt 1):95-105. doi: 10.1042/0264-6021:3510095.

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