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Through the "gatekeeper door": exploiting the active kinase conformation.

作者信息

Zuccotto Fabio, Ardini Elena, Casale Elena, Angiolini Mauro

机构信息

Department of Chemical Core Technologies, Nerviano Medical Sciences, Oncology, Viale Pasteur 10, Nerviano 20014, Italy.

出版信息

J Med Chem. 2010 Apr 8;53(7):2681-94. doi: 10.1021/jm901443h.

DOI:10.1021/jm901443h
PMID:20000735
Abstract
摘要

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