番荔枝环肽B大环的高效合成。
An efficient synthesis of the tamandarin B macrocycle.
作者信息
Lassen Kenneth M, Lee Jisun, Joullié Madeleine M
机构信息
Department of Chemistry, University of Pennsylvania, 231 S. 34 Street, Philadelphia, PA 19104 USA.
出版信息
Tetrahedron Lett. 2010 Mar 31;51(13):1635-1638. doi: 10.1016/j.tetlet.2009.12.091.
Abstract
A reliable, high yielding cyclization protocol for the macrocycle of tamandarin B is presented. This strategy will facilitate the synthesis of side chain analogues.
摘要
本文提出了一种可靠、高产率的环化方案用于合成曼达林B的大环。该策略将有助于侧链类似物的合成。
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