氚标记的（R,R）-4-甲氧基非诺特罗的合成
Synthesis of Tritium Labeled (R,R)-4-Methoxyfenoterol.
作者信息
Kozocas Joseph A, Bupp James E, Tanga Mary J, Pluhar Joseph T, Wainer Irving W
机构信息
SRI International, Menlo Park, CA.
出版信息
J Labelled Comp Radiopharm. 2010 Feb 1;53(2):68-72. doi: 10.1002/jlcr.1703.
Abstract
The preparation of 2',4',6'-[(3)H(3)]-(R,R)-4-methoxyfenoterol, a tritium-labeled derivative of (R,R)-4-methoxyfenoterol was demonstrated on a 15 mCi scale providing material with a specific activity of 57 Ci/mmol.
摘要
制备了2',4',6'-[(3)H(3)]-(R,R)-4-甲氧基非诺特罗，它是(R,R)-4-甲氧基非诺特罗的一种氚标记衍生物，制备规模为15毫居里，得到的产物比活度为57居里/毫摩尔。
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