一锅法合成氮茚类化合物：通过钯催化酮烯醇化物的α-杂芳基化反应。
One-pot synthesis of azaindoles via palladium-catalyzed alpha-heteroarylation of ketone enolates.
机构信息
Bristol-Myers Squibb, Princeton, New Jersey 08543-4000, USA.
出版信息
J Org Chem. 2010 Aug 6;75(15):5316-9. doi: 10.1021/jo100623d.
PMID:20593785
Abstract
A convenient, one-pot method for the construction of a variety of azaindoles using simple ketones and haloaminopyridines is described.
摘要
本文描述了一种简便的一锅法，可利用简单的酮和卤代氨吡啶来构建各种氮茚。
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