γ-氨基丁酸突触拮抗剂[3H]α-二氢印防己毒素与大鼠脑膜的结合。 - Suppr

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超能文献

Binding of [3H]alpha-dihydropicrotoxinin, a gamma-aminobutyric acid synaptic antagonist, to rat brain membranes.

作者信息

Ticku M K, Ban M, Olsen R W

出版信息

Mol Pharmacol. 1978 May;14(3):391-402.

PMID:207968

Abstract

摘要

相似文献

Binding of [3H]alpha-dihydropicrotoxinin, a gamma-aminobutyric acid synaptic antagonist, to rat brain membranes.γ-氨基丁酸突触拮抗剂[3H]α-二氢印防己毒素与大鼠脑膜的结合。

Mol Pharmacol. 1978 May;14(3):391-402.

Dihydropicrotoxinin binding to crayfish muscle sites possibly related to gamma-aminobutyric acid receptor-ionophores.二氢印防己毒素与小龙虾肌肉部位的结合可能与γ-氨基丁酸受体离子载体有关。

Mol Pharmacol. 1978 May;14(3):381-90.

The picrotoxinin binding site and its relationship to the GABA receptor complex.印防己毒素结合位点及其与γ-氨基丁酸受体复合物的关系。

J Neurochem. 1985 Mar;44(3):812-7. doi: 10.1111/j.1471-4159.1985.tb12888.x.

Dihydropicrotoxinin binding sites in rat brain: comparison to GABA receptors.大鼠脑中二氢印防己毒素结合位点：与γ-氨基丁酸受体的比较。

Brain Res. 1978 Jul 21;150(3):642-7. doi: 10.1016/0006-8993(78)90830-2.

Interaction of barbiturates with dihydropicrotoxinin binding sites related to the GABA receptor-ionophore system.巴比妥类药物与二氢印防己毒素结合位点的相互作用，该位点与γ-氨基丁酸（GABA）受体-离子载体系统相关。

Life Sci. 1978 May 8;22(18):1643-51. doi: 10.1016/0024-3205(78)90061-9.

GABA receptor binding and endogenous inhibitors in normal human brain and Huntington's disease.正常人类大脑和亨廷顿舞蹈病中的γ-氨基丁酸（GABA）受体结合与内源性抑制剂

Adv Biochem Psychopharmacol. 1980;21:451-60.

gamma-Aminobutyric acid agonists and antagonists alter chloride flux across brain membranes.γ-氨基丁酸激动剂和拮抗剂会改变氯离子通过脑膜的通量。

Mol Pharmacol. 1986 May;29(5):497-505.

Biochemical identification of the gamma-aminobutyric acid (GABA) receptor in mammalian brain [proceedings].哺乳动物脑中γ-氨基丁酸（GABA）受体的生化鉴定[会议论文集]

Psychopharmacol Bull. 1977 Jan;13(1):29-30.

[3H]alpha-dihydropicrotoxinin binds to primary brain but not to glial cultures.

Eur J Pharmacol. 1980 Jul 11;65(1):135-6. doi: 10.1016/0014-2999(80)90225-3.

Interaction of stereoisomers of barbiturates with [3H]alpha-dihydropicrotoxinin binding sites.

Brain Res. 1981 Apr 27;211(1):127-33. doi: 10.1016/0006-8993(81)90071-8.

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Picrotoxin dramatically speeds the mammalian circadian clock independent of Cys-loop receptors.苦毒蕈碱显著加速哺乳动物生物钟，而不依赖于 Cys 环受体。

J Neurophysiol. 2013 Jul;110(1):103-8. doi: 10.1152/jn.00220.2013. Epub 2013 Apr 10.

Ginkgolide B and bilobalide block the pore of the 5-HT₃receptor at a location that overlaps the picrotoxin binding site.银杏内酯 B 和白果内酯在与苦味酸结合位点重叠的位置阻塞 5-HT₃ 受体的孔。

Neuropharmacology. 2011 Feb-Mar;60(2-3):488-95. doi: 10.1016/j.neuropharm.2010.11.003. Epub 2010 Nov 5.

Structural model for gamma-aminobutyric acid receptor noncompetitive antagonist binding: widely diverse structures fit the same site.γ-氨基丁酸受体非竞争性拮抗剂结合的结构模型：多种不同结构契合同一位点。

Proc Natl Acad Sci U S A. 2006 Mar 28;103(13):5185-90. doi: 10.1073/pnas.0600370103. Epub 2006 Mar 10.

GABA receptor-mediated inhibition of reflex deglutition in the cat.γ-氨基丁酸（GABA）受体介导的对猫反射性吞咽的抑制作用。

Dysphagia. 1996 Summer;11(3):209-15. doi: 10.1007/BF00366388.

Interaction of picrotoxin with GABAA receptor channel-lining residues probed in cysteine mutants.在半胱氨酸突变体中探究印防己毒素与GABAA受体通道内衬残基的相互作用。

Biophys J. 1995 Nov;69(5):1858-67. doi: 10.1016/S0006-3495(95)80056-1.

Multiple mechanisms of picrotoxin block of GABA-induced currents in rat hippocampal neurons.印防己毒素对大鼠海马神经元中γ-氨基丁酸诱导电流的多种阻断机制。

J Physiol. 1993 May;464:423-39. doi: 10.1113/jphysiol.1993.sp019643.

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