新型苯并三唑啉酮衍生物的合成及生物活性。
Synthesis and biological activity of novel phenyltriazolinone derivatives.
机构信息
Key Laboratory of Pesticide and Chemical Biology of Ministry of Education, College of Chemistry, Central China Normal University, Wuhan 430079, Hubei, China.
出版信息
Molecules. 2010 Dec 9;15(12):9024-34. doi: 10.3390/molecules15129024.
Phenyltriazolinones are one of the most important classes of herbicides targeting the protoporphyrinogen oxidase enzyme. A series of triazolinone derivatives containing a strobilurin pharmacophore were designed and synthesized with the aim of discovering new phenyltriazolinone analogues with high activity. The herbicidal activity of the synthesized compounds was assayed and some of the test compounds displayed moderate herbicidal activity at 150 g ai/ha.
苯并三唑酮类是一类最重要的除草剂，作用靶标为原卟啉原氧化酶。为了发现具有高活性的新型苯并三唑酮类似物，设计并合成了一系列含有嘧菌酯药效团的三唑啉酮衍生物。测定了所合成化合物的除草活性，部分测试化合物在 150 g ai/ha 下显示出中等除草活性。
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