Department of Chemistry, Zhejiang University, Hangzhou 310027, P. R. China.
Chem Commun (Camb). 2011 Mar 21;47(11):3275-7. doi: 10.1039/c0cc04922k. Epub 2011 Feb 1.
A three-component reaction of indoles, sulfonyl azides and terminal alkynes afforded 3-functionalized indoles in a single step via copper-cascade catalysis.
吲哚、磺酰叠氮化物和末端炔烃的三组分反应通过铜级联催化一步合成 3 官能化吲哚。