能以选择性和高亲和力与催产素受体结合的受体配体。一种源自淡紫链霉菌的环六肽的化学修饰。 - Suppr | 超能文献

Receptor ligands which bind the oxytocin receptor with selectivity and high affinity. Chemical modification of a Streptomyces silvensis derived cyclic hexapeptide.

作者信息

Bock M G, DiPardo R M, Williams P D, Pettibone D J, Clineschmidt B V, Ball R G, Veber D F, Freidinger R M

机构信息

Department of Medicinal Chemistry, Merck, Sharp & Dohme Research Laboratories, West Point, Pennsylvania 198486.

出版信息

J Med Chem. 1990 Sep;33(9):2321-3. doi: 10.1021/jm00171a003.

DOI:10.1021/jm00171a003

Abstract

摘要

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