Cephalon, Inc., 145 Brandywine Parkway, West Chester, PA 19380-4245, USA.
Bioorg Med Chem Lett. 2012 Mar 15;22(6):2312-4. doi: 10.1016/j.bmcl.2011.12.099. Epub 2011 Dec 29.
In search of a next generation molecule to the novel wake promoting agent modafinil, a series of bi-phenyl derived wakefulness enhancing agents (in rat) was developed. From this work, compound 17 has been selected for additional studies.
为了寻找一种比新型觉醒促进剂莫达非尼更具潜力的下一代分子,我们开发了一系列双苯衍生的觉醒增强剂(在大鼠中)。在这项工作中,化合物 17 被选中进行进一步研究。