Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian 116023, China.
Org Biomol Chem. 2012 Oct 7;10(37):7479-82. doi: 10.1039/c2ob26270c.
Palladium-catalyzed desulfitative and denitrogenative arylation of azoles with arylsulfonyl hydrazides has been achieved. A broad scope of azoles and arylsulfonyl hydrazides has been used to produce arylated azoles in high yields.
钯催化唑类化合物与芳基磺酰基腙的脱硫化和脱氮芳基化反应已经实现。该反应具有广泛的底物适用性,使用各种唑类化合物和芳基磺酰基腙可以高产率得到芳基化唑类化合物。