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Spiperone: a ligand of choice for neuroleptic receptors. 2. Regional distribution and in vivo displacement of neuroleptic drugs.

作者信息

Laduron P M, Janssen P F, Leysen J E

出版信息

Biochem Pharmacol. 1978 Feb 1;27(3):317-21. doi: 10.1016/0006-2952(78)90234-4.

DOI:10.1016/0006-2952(78)90234-4
PMID:23127
Abstract
摘要

相似文献

1
Spiperone: a ligand of choice for neuroleptic receptors. 2. Regional distribution and in vivo displacement of neuroleptic drugs.螺哌隆：一种用于抗精神病药物受体的理想配体。2. 抗精神病药物的区域分布及体内置换
Biochem Pharmacol. 1978 Feb 1;27(3):317-21. doi: 10.1016/0006-2952(78)90234-4.
2
Spiperone: a ligand of choice for neuroleptic receptors. 3. Subcellular distribution of neuroleptic drugs and their receptors in various rat brain areas.螺哌隆：抗精神病药物受体的首选配体。3. 抗精神病药物及其受体在大鼠不同脑区的亚细胞分布。
Biochem Pharmacol. 1978 Feb 1;27(3):323-8. doi: 10.1016/0006-2952(78)90235-6.
3
Spiperone: a ligand of choice for neuroleptic receptors. 1. Kinetics and characteristics of in vitro binding.螺哌隆：一种用于抗精神病药物受体的理想配体。1. 体外结合的动力学和特性
Biochem Pharmacol. 1978 Feb 1;27(3):307-16. doi: 10.1016/0006-2952(78)90233-2.
4
The low affinity component of [3H]spiperone binding reflects association to a non-dopaminergic, neuroleptic site.[3H]司哌罗宁结合的低亲和力成分反映了与非多巴胺能、抗精神病药物位点的结合。
Neurosci Lett. 1982 Apr 16;29(2):147-51. doi: 10.1016/0304-3940(82)90344-5.
5
The effects of standard neuroleptic compounds on the binding of 3H-spiroperidol in the striatum and mesolimbic system of the rat in vitro.标准抗精神病化合物对大鼠纹状体和中脑边缘系统中3H-螺哌啶醇体外结合的影响。
Life Sci. 1978 Aug 14;23(6):599-603. doi: 10.1016/0024-3205(78)90039-5.
6
Regional blockade by neuroleptic drugs of in vivo 3H-spiperone binding in the rat brain. Relation to blockade of apomorphine induced hyperactivity and stereotypies.抗精神病药物对大鼠脑内体内3H-螺哌隆结合的区域阻断作用。与阿扑吗啡诱导的多动和刻板行为阻断的关系。
J Neural Transm. 1981;52(3):163-73. doi: 10.1007/BF01249601.
7
Dopamine receptors in bovine retina : characterization of the 3H-spiroperidol binding and its use for screening dopamine receptor affinity of drugs.
Life Sci. 1979 Nov 5;25(19):1675-86. doi: 10.1016/0024-3205(79)90409-0.
8
Identity and properties of multiple neuroleptic-binding sites in rat limbic brain areas [proceedings].大鼠边缘脑区多个抗精神病药物结合位点的特性与鉴定[会议论文集]
Arch Int Physiol Biochim. 1979 Oct;87(4):822-4.
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Biochemical mechanism of tolerance to neuroleptic drugs; regional differences in rat brain.抗精神病药物耐受性的生化机制；大鼠脑内的区域差异。
Eur J Pharmacol. 1981 Apr 9;70(4):585-6. doi: 10.1016/0014-2999(81)90371-x.
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Similarities and dissimilarities between dopamine and neuroleptic receptors: further evidence for type 1 and type 2 dopamine receptors in the CNS.多巴胺与抗精神病药物受体之间的异同：中枢神经系统中1型和2型多巴胺受体的进一步证据
Adv Biochem Psychopharmacol. 1980;24:113-21.

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In vivo 3H-d-LSD binding in small punched out rat brain regions.
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