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A new selective inhibitor of mouse blood plasma carboxylesterase.

作者信息

Rudakova E V, Makhaeva G F, Galenko T G, Aksinenko A Yu, Sokolov V B, Martynov I V

机构信息

Institute of Physiologically Active Compounds, Russian Academy of Sciences, Chernogolovka, Moscow region, Russia.

出版信息

Dokl Biochem Biophys. 2013 Mar-Apr;449:87-9. doi: 10.1134/S1607672913020099. Epub 2013 May 9.

DOI:10.1134/S1607672913020099
PMID:23657654
Abstract
摘要

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1
A new selective inhibitor of mouse blood plasma carboxylesterase.
Dokl Biochem Biophys. 2013 Mar-Apr;449:87-9. doi: 10.1134/S1607672913020099. Epub 2013 May 9.
2
Carboxylesterase inhibition and potentiation of soman toxicity.羧酸酯酶抑制作用与梭曼毒性的增强
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Structural requirements for the inhibition of human monocyte carboxylesterase by organophosphorus compounds.有机磷化合物对人单核细胞羧酸酯酶抑制作用的结构要求
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[Features of inhibition of butyrylcholinesterase and carboxylesterase hydrolysis of fluoroanhydride esters by beta,beta-diphenylethylphosphonic acid].[β,β-二苯乙基膦酸对氟酐酯的丁酰胆碱酯酶和羧酸酯酶水解的抑制特性]
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In vitro deacetylation studies with isomeric acetamidobiphenyls using selective carboxylesterase inhibitors.使用选择性羧酸酯酶抑制剂对异构乙酰氨基联苯进行的体外脱乙酰化研究。
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Prevention of tolerance to the organophosphorus anticholinesterase paraoxon with carboxylesterase inhibitors.用羧酸酯酶抑制剂预防对有机磷抗胆碱酯酶对氧磷的耐受性。
Biochem Pharmacol. 1998 May 1;55(9):1419-26. doi: 10.1016/s0006-2952(97)00650-3.
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Role of aliesterase in organophosphate poisoning.
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Inhibition of sulphation of phenolic substances by the carboxylesterase inhibitor bis-(p-nitrophenyl)-phosphate in the rat in vivo.大鼠体内羧酸酯酶抑制剂双（对硝基苯基）磷酸酯对酚类物质硫酸化的抑制作用。
Biochem Pharmacol. 1979 Sep 1;28(17):2685-6. doi: 10.1016/0006-2952(79)90051-0.
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The identification and characterization of two separate carboxylesterases in guinea-pig serum.豚鼠血清中两种不同羧酸酯酶的鉴定与特性研究。
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Alkyl 2-arylhydrazinylidene-3-oxo-3-polyfluoroalkylpropionates as new effective and selective inhibitors of carboxylesterase.2-芳基肼叉基-3-氧代-3-多氟烷基丙酸烷基酯作为新型有效的羧酸酯酶选择性抑制剂。
Dokl Biochem Biophys. 2015;465:381-5. doi: 10.1134/S1607672915060101. Epub 2016 Jan 5.

本文引用的文献

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Comparative analysis of esterase activities of human, mouse, and rat blood.人、小鼠和大鼠血液酯酶活性的比较分析。
Bull Exp Biol Med. 2011 Nov;152(1):73-5. doi: 10.1007/s10517-011-1457-y.
2
Production of ES1 plasma carboxylesterase knockout mice for toxicity studies.用于毒性研究的 ES1 血浆羧酸酯酶基因敲除小鼠的生产。
Chem Res Toxicol. 2011 Nov 21;24(11):1891-8. doi: 10.1021/tx200237a. Epub 2011 Sep 7.
3
Carboxylesterase inhibitors.羧酸酯酶抑制剂。
Expert Opin Ther Pat. 2011 Aug;21(8):1159-71. doi: 10.1517/13543776.2011.586339. Epub 2011 May 24.
4
Activity-based protein profiling of organophosphorus and thiocarbamate pesticides reveals multiple serine hydrolase targets in mouse brain.基于活性的有机磷和硫代氨基甲酸酯类农药蛋白质组学分析揭示了小鼠脑中多种丝氨酸水解酶的靶标。
J Agric Food Chem. 2011 Apr 13;59(7):2808-15. doi: 10.1021/jf101747r. Epub 2010 Jul 21.
5
Utility of the carboxylesterase inhibitor bis-para-nitrophenylphosphate (BNPP) in the plasma unbound fraction determination for a hydrolytically unstable amide derivative and agonist of the TGR5 receptor.羧酸酯酶抑制剂双对硝基苯磷酸酯（BNPP）在测定一种水解不稳定的酰胺衍生物及TGR5受体激动剂的血浆游离分数中的应用。
Xenobiotica. 2010 Jun;40(6):369-80. doi: 10.3109/00498251003706598.
6
Improving the ex vivo stability of drug ester compounds in rat and dog serum: inhibition of the specific esterases and implications on their identity.提高药物酯类化合物在大鼠和犬血清中的体外稳定性：抑制特定的酯酶及其对其身份的影响。
J Pharm Biomed Anal. 2010 Feb 5;51(3):664-78. doi: 10.1016/j.jpba.2009.09.023. Epub 2009 Sep 23.
7
Synthesis of organophosphates with fluorine-containing leaving groups as serine esterase inhibitors with potential for Alzheimer disease therapeutics.含氟离去基团的有机磷酸酯作为丝氨酸酯酶抑制剂的合成及其在阿尔茨海默病治疗中的潜力。
Bioorg Med Chem Lett. 2009 Oct 1;19(19):5528-30. doi: 10.1016/j.bmcl.2009.08.065. Epub 2009 Aug 21.
8
Esterase profile and analysis of structure-inhibitor selectivity relationships for homologous phosphorylated 1-hydroperfluoroisopropanols.同源磷酸化1-氢全氟异丙醇的酯酶谱及结构-抑制剂选择性关系分析
Dokl Biochem Biophys. 2008 Nov-Dec;423:352-7. doi: 10.1134/s1607672908060094.
9
Structure and catalytic properties of carboxylesterase isozymes involved in metabolic activation of prodrugs.参与前药代谢活化的羧酸酯酶同工酶的结构与催化特性。
Molecules. 2008 Feb 18;13(2):412-31. doi: 10.3390/molecules13020412.
10
Butyrylcholinesterase, paraoxonase, and albumin esterase, but not carboxylesterase, are present in human plasma.丁酰胆碱酯酶、对氧磷酶和白蛋白酯酶存在于人体血浆中，但羧酸酯酶不存在。
Biochem Pharmacol. 2005 Nov 25;70(11):1673-84. doi: 10.1016/j.bcp.2005.09.002. Epub 2005 Oct 6.