Department of Chemistry, Zhejiang University , Hangzhou 310027, P. R. China.
Org Lett. 2013 Jun 21;15(12):2982-5. doi: 10.1021/ol401144m. Epub 2013 Jun 7.
A concise method for the preparation of tryptanthrins from indoles via the copper-catalyzed aerobic oxidation is described. The reactions can be carried out under mild reaction conditions with varying functional group tolerance.
本文描述了一种通过铜催化的有氧氧化从吲哚类化合物制备色胺酮的简洁方法。该反应可以在温和的反应条件下进行,并具有不同官能团的耐受性。