β-烯胺酯和硫酯的化学选择性合成路线。
A chemoselective route to β-enamino esters and thioesters.
机构信息
Texas A & M University , Chemistry Department, P.O. Box 30012, College Station, Texas 77842, United States.
出版信息
Org Lett. 2014 Apr 18;16(8):2108-10. doi: 10.1021/ol5005643. Epub 2014 Mar 31.
Abstract
Conditions were developed for syntheses of β-enamino esters, thioesters, and amides. These reactions involve hydroxybenzotriazole derivatives in buffered media. Illustrative syntheses of some heterocyclic systems are given, including some related to protein-protein interface mimics.
摘要
本文发展了β-烯胺酯、硫酯和酰胺的合成条件。这些反应涉及缓冲介质中的羟基苯并三唑衍生物。给出了一些杂环体系的示例合成，包括一些与蛋白质-蛋白质界面模拟物相关的合成。
Zotero 插件