[3H]-BRL 43694（格拉司琼），大鼠脑皮质膜中5-HT3结合位点的特异性配体。 - Suppr

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超能文献

[3H]-BRL 43694 (Granisetron), a specific ligand for 5-HT3 binding sites in rat brain cortical membranes.

作者信息

Nelson D R, Thomas D R

机构信息

Beecham Pharmaceuticals Research Division, The Pinnacles Harlow, Essex.

出版信息

Biochem Pharmacol. 1989 May 15;38(10):1693-5. doi: 10.1016/0006-2952(89)90319-5.

DOI:10.1016/0006-2952(89)90319-5

PMID:2543418

Abstract

摘要

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[3H]-BRL 43694 (Granisetron), a specific ligand for 5-HT3 binding sites in rat brain cortical membranes.[3H]-BRL 43694（格拉司琼），大鼠脑皮质膜中5-HT3结合位点的特异性配体。

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Evidence that the atypical 5-HT3 receptor ligand, [3H]-BRL46470, labels additional 5-HT3 binding sites compared to [3H]-granisetron.与[3H] - 格拉司琼相比，非典型5 - HT3受体配体[3H] - BRL46470标记额外5 - HT3结合位点的证据。

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