‡State Key Laboratory of Applied Organic Chemistry, Lanzhou University, Lanzhou 730000, P. R. China.
Org Lett. 2015 Apr 17;17(8):1914-7. doi: 10.1021/acs.orglett.5b00605. Epub 2015 Mar 31.
A multicomponent reaction has been developed for the synthesis of polyfunctional pyrazole derivatives from readily available arylglyoxal monohydrates, tosylhydrazine, and aldehydes or ketones. This synthetic method has significant advantages in broad substrate scope, excellent regioselectivity, and simple operation.
已经开发出一种多组分反应，用于从易得的芳基乙二醛一水合物、对甲苯磺酰肼以及醛或酮合成多功能吡唑衍生物。这种合成方法在广泛的底物范围、优异的区域选择性和简单的操作方面具有显著的优势。
