Lemaire D, Jacob P, Shulgin A T
J Pharm Pharmacol. 1985 Aug;37(8):575-7. doi: 10.1111/j.2042-7158.1985.tb03072.x.
Four members of a new class of psychotomimetic agents have been synthesized and evaluated in man. These compounds, which incorporate a beta-methoxy group onto a beta-phenethylamine sidechain, are the first reported psychotomimetics which are structural analogues of the neurotransmitter noradrenaline. These substances are more potent than the corresponding phenethylamines (lacking a beta-methoxy group) but less potent than the correspondingly substituted amphetamine derivatives.
