咪唑化合物作为组胺甲基转移酶抑制剂或激活剂的结构要求：组胺类似物和H2受体拮抗剂的研究 - Suppr

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Structural requirements of imidazole compounds to be inhibitors or activators of histamine methyltransferase: investigation of histamine analogues and H2-receptor antagonists.

作者信息

Barth H, Lorenz W

出版信息

Agents Actions. 1978 Jun;8(4):359-65. doi: 10.1007/BF01968615.

DOI:10.1007/BF01968615

PMID:28646

Abstract

摘要

相似文献

Structural requirements of imidazole compounds to be inhibitors or activators of histamine methyltransferase: investigation of histamine analogues and H2-receptor antagonists.咪唑化合物作为组胺甲基转移酶抑制剂或激活剂的结构要求：组胺类似物和H2受体拮抗剂的研究

Agents Actions. 1978 Jun;8(4):359-65. doi: 10.1007/BF01968615.

Evidence for a less high acceptor substrate specificity of gastric histamine methyltransferase: methylation of imidazole compounds.胃组胺甲基转移酶受体底物特异性较低的证据：咪唑化合物的甲基化

Biochem Pharmacol. 1980 May 15;29(10):1399-407. doi: 10.1016/0006-2952(80)90436-0.

Sidechain-modified histamine analogues as substrates for histamine N-methyltransferase.作为组胺N-甲基转移酶底物的侧链修饰组胺类似物

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Bioisosteric prototype design of biaryl imidazolyl and triazolyl competitive histamine H2-receptor antagonists.联芳基咪唑基和三唑基竞争性组胺H2受体拮抗剂的生物电子等排体原型设计

J Med Chem. 1986 Nov;29(11):2154-63. doi: 10.1021/jm00161a005.

Pharmacological properties of histamine-sensitive adenylate cyclase from mammalian brain.哺乳动物脑内组胺敏感腺苷酸环化酶的药理学特性

J Pharmacol Exp Ther. 1979 Apr;209(1):87-96.

Pharmacological properties of histamine-sensitive adenylate cyclase from guinea pig cardiac ventricular muscle.豚鼠心室肌组胺敏感腺苷酸环化酶的药理学特性

Mol Pharmacol. 1979 May;15(3):445-61.

Studies on the mode of action of histamine H1- and H2-receptor antagonists on gastric histamine methyltransferase.组胺H1和H2受体拮抗剂对胃组胺甲基转移酶作用模式的研究。

Agents Actions. 1973 Oct;3(3):138-47. doi: 10.1007/BF01965724.

New inhibitors of histamine-N-methyltransferase.组胺-N-甲基转移酶的新型抑制剂

Biochem Pharmacol. 1979;28(2):183-8. doi: 10.1016/0006-2952(79)90500-8.

Impromidine, a potent inhibitor of histamine methyltransferase (HMT) and diamine oxidase (DAO).英普咪定，一种组胺甲基转移酶（HMT）和二胺氧化酶（DAO）的强效抑制剂。

Biochem Pharmacol. 1980 Oct 15;29(20):2897-900. doi: 10.1016/0006-2952(80)90033-7.

Inhibition and activation of histamine methyltransferase by methylated histamines.甲基化组胺对组胺甲基转移酶的抑制与激活作用

Hoppe Seylers Z Physiol Chem. 1973 Sep;354(9):1021-6. doi: 10.1515/bchm2.1973.354.2.1021.

引用本文的文献

Dual role of imidazole as activator/inhibitor of sweet almond () β-glucosidase.咪唑作为甜杏仁（）β-葡萄糖苷酶激活剂/抑制剂的双重作用。（注：括号内“（）”处原文似乎信息不完整）

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Histamine N-methyltransferase: inhibition by monoamine oxidase inhibitors.组胺N-甲基转移酶：单胺氧化酶抑制剂的抑制作用

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Inhibition of plant and mammalian diamine oxidase by substrate analogues.底物类似物对植物和哺乳动物二胺氧化酶的抑制作用。

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Gastric histamine methyltransferase: different methylation rates for enantiomers of side-chain methylated histamine analogues using a highly purified enzyme preparation.胃组胺甲基转移酶：使用高度纯化的酶制剂对侧链甲基化组胺类似物对映体的不同甲基化率。

Agents Actions. 1984 Apr;14(3-4):346-50. doi: 10.1007/BF01973824.

Histamine uptake and metabolism in intact isolated parietal cells.完整分离壁细胞中的组胺摄取与代谢

Agents Actions. 1981 May;11(3):223-7. doi: 10.1007/BF01967618.

H1 + H2-receptor antagonists for premedication in anaesthesia and surgery: a critical view based on randomized clinical trials with Haemaccel and various antiallergic drugs.用于麻醉和手术术前用药的H1+H2受体拮抗剂：基于使用贺斯（Haemaccel）和各种抗过敏药物的随机临床试验的批判性观点

Agents Actions. 1980 Apr;10(1 Pt 2):114-24. doi: 10.1007/BF02024192.

Inhibition of histamine-N-methyltransferase activity by neuromuscular blocking drugs.神经肌肉阻滞药物对组胺-N-甲基转移酶活性的抑制作用。

Agents Actions. 1985 Oct;17(1):27-31. doi: 10.1007/BF01966676.

Histamine N-methyl transferase: inhibition by drugs.组胺N-甲基转移酶：药物抑制作用

Br J Clin Pharmacol. 1992 Oct;34(4):322-7. doi: 10.1111/j.1365-2125.1992.tb05637.x.

Inhibition of histamine methylation in vivo by the dimaprit analog, SKF Compound 91488.地马普利类似物SKF化合物91488对体内组胺甲基化的抑制作用。

Agents Actions. 1979 Dec;9(5-6):455-60. doi: 10.1007/BF01968110.

本文引用的文献

Protein measurement with the Folin phenol reagent.使用福林酚试剂进行蛋白质测定。

J Biol Chem. 1951 Nov;193(1):265-75.

Biochem Pharmacol. 1980 May 15;29(10):1399-407. doi: 10.1016/0006-2952(80)90436-0.

Sex differences and hormonal control of histamine methyltransferase activity.组胺甲基转移酶活性的性别差异与激素调控

Biochim Biophys Acta. 1965 Dec 16;111(2):416-21. doi: 10.1016/0304-4165(65)90051-6.

Inhibition and activation of histamine methyltransferase by methylated histamines.甲基化组胺对组胺甲基转移酶的抑制与激活作用

Hoppe Seylers Z Physiol Chem. 1973 Sep;354(9):1021-6. doi: 10.1515/bchm2.1973.354.2.1021.

A sensitive and specific method for the determination of histomine in human whole blood and plasma.一种测定人全血和血浆中组胺的灵敏且特异的方法。

Hoppe Seylers Z Physiol Chem. 1972 Jun;353(6):911-20. doi: 10.1515/bchm2.1972.353.1.911.

Speculations about the binding sites of S-adenosyl-L-homocysteine and some of its synthetic analogues to histamine methyltransferase.关于S-腺苷-L-同型半胱氨酸及其一些合成类似物与组胺甲基转移酶结合位点的推测。

Agents Actions. 1974 Aug;4(3):186-8. doi: 10.1007/BF01970266.

Histamine methyltransferase: inhibition and potentiation by antihistamines.组胺甲基转移酶：抗组胺药对其的抑制与增强作用

Mol Pharmacol. 1972 May;8(3):300-10.

Definition and antagonism of histamine H 2 -receptors.组胺H2受体的定义与拮抗作用。

Nature. 1972 Apr 21;236(5347):385-90. doi: 10.1038/236385a0.

Sulphur-methylene isosterism in the development of metiamide, a new histamine H2-receptor antagonist.新型组胺H2受体拮抗剂甲硫米特研发中的硫-亚甲基电子等排原理

Nature. 1974 Mar 1;248(5443):65-7. doi: 10.1038/248065a0.

Agents Actions. 1973 Oct;3(3):173-5. doi: 10.1007/BF01965730.

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