Quazepam, a sedative-hypnotic selective for the benzodiazepine type 1 receptor: autoradiographic localization in rat and human brain.
作者信息
Wamsley J K, Golden J S, Yamamura H I, Barnett A
出版信息
Clin Neuropharmacol. 1985;8 Suppl 1:S26-40. doi: 10.1097/00002826-198508001-00005.
Abstract
摘要
相似文献
1
Quazepam, a sedative-hypnotic selective for the benzodiazepine type 1 receptor: autoradiographic localization in rat and human brain.夸西泮，一种对苯二氮䓬1型受体有选择性的镇静催眠药：在大鼠和人类大脑中的放射自显影定位。
Clin Neuropharmacol. 1985;8 Suppl 1:S26-40. doi: 10.1097/00002826-198508001-00005.
2
Autoradiographic demonstration of the selectivity of two 1-N-trifluoroethyl benzodiazepines for the BZD-1 receptors in the rat brain.
Pharmacol Biochem Behav. 1985 Dec;23(6):973-8. doi: 10.1016/0091-3057(85)90103-0.
3
Relative affinity of quazepam for type-1 benzodiazepine receptors in brain.
J Clin Psychiatry. 1991 Sep;52 Suppl:15-20.
4
Use of the selective benzodiazepine-1 (BZ-1) ligand [3H]2-oxo-quazepam (SCH 15-725) to localize BZ-1 receptors in the rat brain.
Neurosci Lett. 1988 May 16;88(1):86-92. doi: 10.1016/0304-3940(88)90320-5.
5
6
Selective affinity of the benzodiazepines quazepam and 2-oxo-quazepam for BZ1 binding site and demonstration of 3H-2-oxo-quazepam as a BZ1 selective radioligand.苯二氮䓬类药物夸西泮和2-氧代夸西泮对BZ1结合位点的选择性亲和力以及3H-2-氧代夸西泮作为BZ1选择性放射性配体的证明。
Life Sci. 1988;42(2):179-87. doi: 10.1016/0024-3205(88)90681-9.
7
Contribution of specific binding to the central benzodiazepine site to the brain concentrations of two novel benzodiazepine site ligands.特异性结合至中枢苯二氮䓬位点对两种新型苯二氮䓬位点配体脑内浓度的贡献。
Biopharm Drug Dispos. 2007 Sep;28(6):275-82. doi: 10.1002/bdd.553.
8
Several new benzodiazepines selectively interact with a benzodiazepine receptor subtype.
Neurosci Lett. 1983 Jul 15;38(1):73-8. doi: 10.1016/0304-3940(83)90113-1.
9
N3-phenacyluridine, a novel hypnotic compound, interacts with the benzodiazepine receptor.N3-苯甲酰基尿苷，一种新型催眠化合物，与苯二氮䓬受体相互作用。
Eur J Pharmacol. 1996 Sep 12;311(2-3):265-9. doi: 10.1016/0014-2999(96)00434-7.
10
High affinity inhibition of [3H]-flunitrazepam binding to brain benzodiazepine receptors by CGS 9896, a novel pyrazoloquinoline.
Biochem Biophys Res Commun. 1982 Mar 30;105(2):457-61. doi: 10.1016/0006-291x(82)91456-5.
引用本文的文献
1
Quazepam. A preliminary review of its pharmacodynamic and pharmacokinetic properties, and therapeutic efficacy in insomnia.夸西泮。对其药效学和药代动力学特性以及在失眠治疗中的疗效的初步综述。
Drugs. 1988 Jan;35(1):42-62. doi: 10.2165/00003495-198835010-00003.
Zotero 插件