[3H]CPP，一种新型的NMDA受体竞争性配体。 - Suppr

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[3H]CPP, a new competitive ligand for NMDA receptors.

作者信息

Olverman H J, Monaghan D T, Cotman C W, Watkins J C

出版信息

Eur J Pharmacol. 1986 Nov 12;131(1):161-2. doi: 10.1016/0014-2999(86)90533-9.

DOI:10.1016/0014-2999(86)90533-9

PMID:3028828

Abstract

摘要

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[3H]CPP, a new competitive ligand for NMDA receptors.[3H]CPP，一种新型的NMDA受体竞争性配体。

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CPP, a selective N-methyl-D-aspartate (NMDA)-type receptor antagonist: characterization in vitro and in vivo.CPP，一种选择性N-甲基-D-天冬氨酸（NMDA）型受体拮抗剂：体内外特性研究

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Evidence for a functional coupling of the NMDA and glycine recognition sites in synaptic plasma membranes.突触质膜中NMDA和甘氨酸识别位点功能偶联的证据。

Eur J Pharmacol. 1990 Jan 23;188(1):63-70. doi: 10.1016/0922-4106(90)90248-v.

Radioligand labeling of N-methyl-D-aspartic acid (NMDA) receptors by [3H](+-)-3-(2-carboxypiperazin-4-yl)propyl-1-phosphonic acid in brain synaptic membranes treated with Triton X-100.用[3H](+-)-3-(2-羧基哌嗪-4-基)丙基-1-膦酸对经Triton X-100处理的脑突触膜中的N-甲基-D-天冬氨酸（NMDA）受体进行放射性配体标记。

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The novel anticonvulsant MK-801 binds to the activated state of the N-methyl-D-aspartate receptor in rat brain.新型抗惊厥药MK-801与大鼠脑中N-甲基-D-天冬氨酸受体的激活状态相结合。

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Characterization of organophosphate interactions at N-methyl-D-aspartate receptors in brain synaptic membranes.脑突触膜中N-甲基-D-天冬氨酸受体上有机磷酸酯相互作用的表征

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Guanine nucleotide modulation of [3H]TCP binding to the NMDA receptor complex.

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Glutamine mimics glycine to enhance [3H]TCP binding at the NMDA receptor complex.

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[3H]glycine binding is modulated by Mg2+ and other ligands of the NMDA receptor-cation channel complex.[3H]甘氨酸结合受Mg2+以及N-甲基-D-天冬氨酸受体-阳离子通道复合物的其他配体调节。

Eur J Pharmacol. 1988 Jun 22;151(1):157-8. doi: 10.1016/0014-2999(88)90709-1.

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Stimulation of serotonin release in the rat brain cortex by activation of ionotropic glutamate receptors and its modulation via alpha 2-heteroreceptors.离子型谷氨酸受体激活对大鼠大脑皮层5-羟色胺释放的刺激作用及其通过α2异受体的调节

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A comparison between the in vivo and in vitro activity of five potent and competitive NMDA antagonists.五种强效竞争性N-甲基-D-天冬氨酸拮抗剂的体内和体外活性比较。

Br J Pharmacol. 1988 Nov;95(3):957-65. doi: 10.1111/j.1476-5381.1988.tb11726.x.

Two classes of N-methyl-D-aspartate recognition sites: differential distribution and differential regulation by glycine.两类N-甲基-D-天冬氨酸识别位点：甘氨酸的差异分布与差异调节

Proc Natl Acad Sci U S A. 1988 Dec;85(24):9836-40. doi: 10.1073/pnas.85.24.9836.

3H-labeled MK-801 binding to the excitatory amino acid receptor complex from rat brain is enhanced by glycine.甘氨酸可增强3H标记的MK-801与大鼠脑兴奋性氨基酸受体复合物的结合。

Proc Natl Acad Sci U S A. 1987 Nov;84(21):7744-8. doi: 10.1073/pnas.84.21.7744.

CGP 37849 and CGP 39551: novel and potent competitive N-methyl-D-aspartate receptor antagonists with oral activity.CGP 37849和CGP 39551：新型强效竞争性N-甲基-D-天冬氨酸受体拮抗剂，具有口服活性。

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The pharmacological specificity of N-methyl-D-aspartate receptors in rat cerebral cortex: correspondence between radioligand binding and electrophysiological measurements.大鼠大脑皮层中 N-甲基-D-天冬氨酸受体的药理学特异性：放射性配体结合与电生理测量之间的对应关系。

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