吗啡 - 6 - 葡萄糖醛酸对阿片受体具有高亲和力。 - Suppr

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超能文献

Morphine-6-glucuronide has high affinity for the opioid receptor.

作者信息

Christensen C B, Jørgensen L N

出版信息

Pharmacol Toxicol. 1987 Jan;60(1):75-6. doi: 10.1111/j.1600-0773.1987.tb01724.x.

DOI:10.1111/j.1600-0773.1987.tb01724.x

PMID:3031640

Abstract

摘要

相似文献

Morphine-6-glucuronide has high affinity for the opioid receptor.吗啡 - 6 - 葡萄糖醛酸对阿片受体具有高亲和力。

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14 beta-(Bromoacetamido)morphine irreversibly labels mu opioid receptors in rat brain membranes.14-β-（溴乙酰胺基）吗啡不可逆地标记大鼠脑膜中的μ阿片受体。

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Explanation at the opioid receptor level for differing toxicity of morphine and morphine 6-glucuronide.吗啡和吗啡-6-葡萄糖醛酸苷不同毒性在阿片受体水平的解释。

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The opiate receptor.阿片受体。

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Morphine-6-glucuronide is more mu-selective and potent in analgesic tests than morphine.吗啡 -6-葡萄糖醛酸在镇痛试验中比吗啡具有更高的μ受体选择性和更强的效力。

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A comparative study of the effect of methionine enkephalin upon the stereospecific binding of an opiate agonist and an antagonist in mice and rats.

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[The role of morphine-6-glucuronide during longterm administration of morphine.].

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Blood-brain barrier transport and brain distribution of morphine-6-glucuronide in relation to the antinociceptive effect in rats--pharmacokinetic/pharmacodynamic modelling.吗啡-6-葡萄糖醛酸苷的血脑屏障转运及脑内分布与大鼠抗伤害感受作用的关系——药代动力学/药效学建模

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