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双吡唑酮:小麦中新的 HPPD 抑制剂除草剂。

Bipyrazone: a new HPPD-inhibiting herbicide in wheat.

机构信息

College of Plant Protection, Shandong Agricultural University, Tai'an, 271018, Shandong, P.R. China.

Key Laboratory of Pesticide Toxicology and Application Technique, College of Plant Protection, Shandong Agricultural University, Tai'an, 271018, Shandong, P.R. China.

出版信息

Sci Rep. 2020 Mar 26;10(1):5521. doi: 10.1038/s41598-020-62116-6.

DOI:10.1038/s41598-020-62116-6
PMID:32218463
原文链接:https://pmc.ncbi.nlm.nih.gov/articles/PMC7098957/
Abstract

Bipyrazone, 1,3-dimethyl-4-(2-(methylsulfonyl)-4-(trifluoromethyl) benzoyl)-1H-pyrazol-5-yl 1,3-dimethyl-1H-pyrazole- 4-carboxylate, is a 4-hydroxyphenylpyaunate dioxygenase (HPPD)-inhibiting herbicide. Greenhouse and field experiments were conducted to explore the potential of post-emergence (POST) application of bipyrazone in wheat fields in China. In the greenhouse study, bipyrazone at 10 and 20 g active ingredient (a.i.) ha effectively controlled Descurainia sophia L., Capsella bursa-pastoris (L.) Medic., Lithospermum arvense L. and Myosoton aquaticum L. Whereas, all tested 16 wheat cultivars showed high degree of tolerance to bipyrazone at 375 and 750 g a.i. ha. In a dose-response experiment carried on the Shannong 6 wheat cultivar and five weed biotypes, bipyrazone was safe to the wheat cultivar, and C. bursa-pastoris, M. aquaticum and D. sophia were sensitive to this herbicide. The selectivity index (SI) between the Shannong 6 and weeds ranged from 34 to 39. The field experiments confirmed that a mixture of bipyrazone and fluroxypyr-mepthyl is practical for controlling broadleaf weeds, and bipyrazone applied alone at 30 to 40 g a.i. ha can also provide satisfactory control of sensitive broadleaf weeds. These findings suggest that bipyrazone POST application has good potential for broadleaf weed management in wheat fields.

摘要

双吡唑酮,1,3-二甲基-4-[2-(甲基磺酰基)-4-(三氟甲基)苯甲酰基]-1H-吡唑-5-基-1,3-二甲基-1H-吡唑-4-羧酸酯,是一种 4-羟基苯基丙酮酸双加氧酶(HPPD)抑制剂除草剂。本研究通过温室和田间试验,探索了双吡唑酮在我国麦田苗后(POST)应用的潜力。温室研究表明,10 和 20 g a.i.ha 的双吡唑酮可有效防除播娘蒿、荠、猪殃殃和水芹;而 16 个供试小麦品种对 375 和 750 g a.i.ha 的双吡唑酮均表现出高度耐性。在对山农 6 小麦品种和 5 种杂草生物型的剂量反应试验中,双吡唑酮对小麦品种安全,而荠、水芹和播娘蒿对该除草剂敏感。山农 6 与杂草之间的选择性指数(SI)范围为 34 至 39。田间试验证实,双吡唑酮与氟氯吡啶酯的混合物可有效防除阔叶杂草,单独使用 30 至 40 g a.i.ha 的双吡唑酮也能有效防除敏感阔叶杂草。这些发现表明,双吡唑酮 POST 应用具有在麦田中防治阔叶杂草的良好潜力。

https://cdn.ncbi.nlm.nih.gov/pmc/blobs/94ff/7098957/9c40807a0a48/41598_2020_62116_Fig3_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/94ff/7098957/64afd02b732d/41598_2020_62116_Fig1_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/94ff/7098957/c5be0b7fb772/41598_2020_62116_Fig2_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/94ff/7098957/9c40807a0a48/41598_2020_62116_Fig3_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/94ff/7098957/64afd02b732d/41598_2020_62116_Fig1_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/94ff/7098957/c5be0b7fb772/41598_2020_62116_Fig2_HTML.jpg
https://cdn.ncbi.nlm.nih.gov/pmc/blobs/94ff/7098957/9c40807a0a48/41598_2020_62116_Fig3_HTML.jpg

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