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A 5-HT receptor in the central nervous system, positively coupled with adenylate cyclase, is antagonized by ICS 205 930.

作者信息

Dumuis A, Bouhelal R, Sebben M, Bockaert J

机构信息

Centre CNRS-INSERM de Pharmacologie-Endocrinologie, Montpellier, France.

出版信息

Eur J Pharmacol. 1988 Jan 27;146(1):187-8. doi: 10.1016/0014-2999(88)90503-1.

DOI:10.1016/0014-2999(88)90503-1
PMID:3350057
Abstract
摘要

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1
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BRL 24924: a potent agonist at a non-classical 5-HT receptor positively coupled with adenylate cyclase in colliculi neurons.BRL 24924：一种对非经典5-羟色胺受体有强效激动作用的物质，该受体在丘脑中的神经元中与腺苷酸环化酶正性偶联。
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Neuroscientist. 2016 Feb;22(1):26-45. doi: 10.1177/1073858414561303. Epub 2014 Dec 8.
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Synthesis and structure-affinity relationships of selective high-affinity 5-HT(4) receptor antagonists: application to the design of new potential single photon emission computed tomography tracers.选择性高亲和力 5-HT(4) 受体拮抗剂的合成与结构亲和力关系：在新型单光子发射计算机断层扫描示踪剂设计中的应用。
J Med Chem. 2012 Nov 26;55(22):9693-707. doi: 10.1021/jm300943r. Epub 2012 Nov 9.
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Serotonin receptors in hippocampus.
海马体中的血清素受体。
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Poster communications.壁报交流
Br J Pharmacol. 1993 Oct;110(Suppl):81P-184P. doi: 10.1111/j.1476-5381.1993.tb16292.x.
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5-hydroxytryptamine 4 receptor activation of the extracellular signal-regulated kinase pathway depends on Src activation but not on G protein or beta-arrestin signaling.细胞外信号调节激酶途径的5-羟色胺4受体激活依赖于Src激活，而非G蛋白或β-抑制蛋白信号传导。
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Br J Pharmacol. 2001 Apr;132(8):1799-808. doi: 10.1038/sj.bjp.0703988.
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Pharmacological characterization of the 5-hydroxytryptamine receptor mediating relaxation in the rat isolated ileum.介导大鼠离体回肠舒张的5-羟色胺受体的药理学特性
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