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Diketopiperazine derivatives, a new series of platelet-activating factor inhibitors.

作者信息

Shimazaki N, Shima I, Hemmi K, Tsurumi Y, Hashimoto M

出版信息

Chem Pharm Bull (Tokyo). 1987 Aug;35(8):3527-30. doi: 10.1248/cpb.35.3527.

DOI:10.1248/cpb.35.3527
PMID:3427732
Abstract
摘要

相似文献

1
Diketopiperazine derivatives, a new series of platelet-activating factor inhibitors.二酮哌嗪衍生物,一类新型血小板活化因子抑制剂。
Chem Pharm Bull (Tokyo). 1987 Aug;35(8):3527-30. doi: 10.1248/cpb.35.3527.
2
PAF inhibitory activity of diketopiperazines: structure-activity relationships.
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PAF inhibitors of microbial origin. Studies on diketopiperazine derivatives.微生物来源的血小板活化因子(PAF)抑制剂。对二酮哌嗪衍生物的研究。
Prog Biochem Pharmacol. 1988;22:66-80.
4
Synthesis and platelet-activating factor (PAF)-antagonistic activities of 1,4-disubstituted piperazine derivatives.1,4-二取代哌嗪衍生物的合成及其血小板活化因子(PAF)拮抗活性
Chem Pharm Bull (Tokyo). 1994 Mar;42(3):541-50. doi: 10.1248/cpb.42.541.
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Diketopiperazines as a new class of platelet-activating factor inhibitors.二酮哌嗪作为一类新型血小板活化因子抑制剂。
J Med Chem. 1987 Oct;30(10):1706-9. doi: 10.1021/jm00393a002.
6
Synthesis and platelet-activating factor (PAF)-antagonistic activities of trisubstituted piperazine derivatives.三取代哌嗪衍生物的合成及其血小板活化因子(PAF)拮抗活性
Chem Pharm Bull (Tokyo). 1994 Mar;42(3):551-9. doi: 10.1248/cpb.42.551.
7
Synthesis and in vitro evaluation of a series of diketopiperazine inhibitors of plasminogen activator inhibitor-1.一系列纤溶酶原激活物抑制剂-1二酮哌嗪抑制剂的合成与体外评价
Bioorg Med Chem Lett. 2001 Oct 8;11(19):2589-92. doi: 10.1016/s0960-894x(01)00508-x.
8
Structure-activity relationships in platelet-activating factor. Part 14: synthesis and biological evaluation of piperazine derivatives with dual anti-PAF and anti-HIV-1 activity.
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Dual antagonists of platelet activating factor and histamine. 3. Synthesis, biological activity and conformational implications of substituted N-acyl-bis-arylcycloheptapiperazines.血小板活化因子和组胺的双重拮抗剂。3. 取代的N-酰基-双-芳基环庚哌嗪的合成、生物活性及构象意义
Bioorg Med Chem Lett. 1998 Dec 15;8(24):3469-74. doi: 10.1016/s0960-894x(98)00626-x.
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Novel inhibitors of plasminogen activator inhibitor-1: development of new templates from diketopiperazines.纤溶酶原激活物抑制剂-1的新型抑制剂:基于二酮哌嗪开发新模板
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