Open Biol. 2024 Jun;14(6):230272. doi: 10.1098/rsob.230272. Epub 2024 Jun 19.
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Chemical Synthesis and Biological Evaluation of 3-Substituted Estrone/Estradiol Derivatives as 17β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors Acting via a Reverse Orientation of the Natural Substrate Estrone.