硫霉素对大肠杆菌转肽酶活性的抑制作用。
Inhibition of transpeptidase activity in Escherichia coli by thienamycin.
作者信息
Moore B A, Jevons S, Brammer K W
出版信息
Antimicrob Agents Chemother. 1979 Jun;15(6):831-3. doi: 10.1128/AAC.15.6.831.
Abstract
Thienamycin was shown to be a more potent inhibitor than ampicillin of the enzyme peptidoglycan transpeptidase from Escherichia coli.
摘要
研究表明，与氨苄青霉素相比，硫霉素是大肠杆菌肽聚糖转肽酶更有效的抑制剂。
相似文献
1
Inhibition of transpeptidase activity in Escherichia coli by thienamycin.硫霉素对大肠杆菌转肽酶活性的抑制作用。
Antimicrob Agents Chemother. 1979 Jun;15(6):831-3. doi: 10.1128/AAC.15.6.831.
2
Peptidoglycan transpeptidase inhibition in Pseudomonas aeruginosa and Escherichia coli by Penicillins and Cephalosporins.青霉素和头孢菌素对铜绿假单胞菌和大肠杆菌中肽聚糖转肽酶的抑制作用。
Antimicrob Agents Chemother. 1979 Apr;15(4):513-7. doi: 10.1128/AAC.15.4.513.
3
Inhibition of peptidoglycan transpeptidase by beta-lactam antibiotics: structure-activity relationships.β-内酰胺类抗生素对肽聚糖转肽酶的抑制作用：构效关系
J Antibiot (Tokyo). 1980 Nov;33(11):1357-62. doi: 10.7164/antibiotics.33.1357.
4
5-Carboxytetramethylrhodamine-Ampicillin Fluorescence Anisotropy-Based Assay of Escherichia coli Penicillin-Binding Protein 2 Transpeptidase Inhibition.基于5-羧基四甲基罗丹明-氨苄青霉素荧光各向异性的大肠杆菌青霉素结合蛋白2转肽酶抑制测定法
ACS Infect Dis. 2019 Jun 14;5(6):863-872. doi: 10.1021/acsinfecdis.8b00351. Epub 2019 Mar 19.
5
Effect of demycarosylturimycin on ribosomal peptidyltransferase from Escherichia coli.
J Antibiot (Tokyo). 1978 Jun;31(6):610-5. doi: 10.7164/antibiotics.31.610.
6
Lytic response of Escherichia coli cells to inhibitors of penicillin-binding proteins 1a and 1b as a timed event related to cell division.大肠杆菌细胞对青霉素结合蛋白1a和1b抑制剂的裂解反应作为与细胞分裂相关的定时事件。
J Bacteriol. 1989 Aug;171(8):4217-21. doi: 10.1128/jb.171.8.4217-4221.1989.
7
High-throughput screen for inhibitors of transglycosylase and/or transpeptidase activities of Escherichia coli penicillin binding protein 1b.针对大肠杆菌青霉素结合蛋白1b的转糖基酶和/或转肽酶活性抑制剂的高通量筛选。
Antimicrob Agents Chemother. 2004 Jan;48(1):30-40. doi: 10.1128/AAC.48.1.30-40.2004.
8
The effect of ribosomal peptidyl-transferase inhibitors is antagonized by elongation factor G with GTP.核糖体肽基转移酶抑制剂的作用被带有鸟苷三磷酸（GTP）的延伸因子G所拮抗。
FEBS Lett. 1976 Nov;70(1):101-4. doi: 10.1016/0014-5793(76)80735-1.
9
Effect of the leucomycin-like macrolide antibiotic turimycin on ribosomal peptidyltransferase from Eschericha coli.
J Antibiot (Tokyo). 1976 Dec;29(12):1314-7. doi: 10.7164/antibiotics.29.1314.
10
Effect of 7-alpha methoxy substitution of cephalosporins upon their affinity for the penicillin-binding proteins of E. coli K12. Comparison with antibacterial activity and inhibition of membrane bound model transpeptidase activity.头孢菌素7-α甲氧基取代对其与大肠杆菌K12青霉素结合蛋白亲和力的影响。与抗菌活性及膜结合模型转肽酶活性抑制作用的比较。
J Antimicrob Chemother. 1979 Jul;5(4):391-8. doi: 10.1093/jac/5.4.391.
本文引用的文献
1
Protein measurement with the Folin phenol reagent.使用福林酚试剂进行蛋白质测定。
J Biol Chem. 1951 Nov;193(1):265-75.
2
3
Mechanism of action of penicillins: a proposal based on their structural similarity to acyl-D-alanyl-D-alanine.青霉素的作用机制：基于其与酰基-D-丙氨酰-D-丙氨酸结构相似性的一种假说
Proc Natl Acad Sci U S A. 1965 Oct;54(4):1133-41. doi: 10.1073/pnas.54.4.1133.
4
Penicillin: its basic site of action as an inhibitor of a peptide cross-linking reaction in cell wall mucopeptide synthesis.青霉素：其作为细胞壁粘肽合成中肽交联反应抑制剂的基本作用位点。
Proc Natl Acad Sci U S A. 1965 Jul;54(1):75-81. doi: 10.1073/pnas.54.1.75.
5
In vivo and in vitro action of new antibiotics interfering with the utilization of N-acetyl-glucosamine-N-acetyl-muramyl-pentapeptide.干扰N-乙酰葡糖胺-N-乙酰胞壁酰五肽利用的新型抗生素的体内和体外作用
J Bacteriol. 1971 Oct;108(1):20-9. doi: 10.1128/jb.108.1.20-29.1971.
6
7
Interaction of penicillin with the bacterial cell: penicillin-binding proteins and penicillin-sensitive enzymes.青霉素与细菌细胞的相互作用：青霉素结合蛋白和青霉素敏感酶。
Bacteriol Rev. 1974 Sep;38(3):291-335. doi: 10.1128/br.38.3.291-335.1974.
8
The interplay of beta-lactamases and intrinsic factors in the resistance of gram-negative bacteria to penicillins and cephalosporins.β-内酰胺酶与内在因素在革兰氏阴性菌对青霉素和头孢菌素耐药性中的相互作用。
Ann N Y Acad Sci. 1974 May 10;235(0):553-68. doi: 10.1111/j.1749-6632.1974.tb43290.x.
9
Peptidoglycan biosynthesis in a thermosensitive division mutant of Escherichia coli.
Biochemistry. 1976 May 4;15(9):1781-90. doi: 10.1021/bi00654a001.
10
In vitro activity of thienamycin.硫霉素的体外活性。
Antimicrob Agents Chemother. 1978 Sep;14(3):436-8. doi: 10.1128/AAC.14.3.436.
Zotero 插件