Jani M D, Srinivasan S
Indian J Physiol Pharmacol. 1977 Apr-Jun;21(2):159-62.
2-methyl-3(3'-methyl-2'-pyridyl)-4 (3H) quinazolinone (SRC-820) and methaqualone inhibited the growth of Streptococcus faecalis-R (ATCC-8043). Phosphoenolpyruvate formation from 3-phosphoglycerate by an enzyme extract of S. faecalis was inhibited by SRC-820. With edetate or fluoride, an additive inhibitory effect by SRC-820 was observed.
2-甲基-3(3'-甲基-2'-吡啶基)-4(3H)喹唑啉酮(SRC-820)和甲喹酮抑制粪肠球菌-R(ATCC-8043)的生长。SRC-820抑制了粪肠球菌的酶提取物将3-磷酸甘油酸转化为磷酸烯醇丙酮酸的过程。在有依地酸盐或氟化物存在的情况下,观察到SRC-820具有相加抑制作用。