Functional evidence for a second binding site of nicotinic antagonists using phencyclidine derivatives.

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作者信息

Kloog Y, Gabrialevitz A, Kalir A, Balderman D, Sokolovsky M

出版信息

Biochem Pharmacol. 1979 Apr 15;28(8):1447-50. doi: 10.1016/0006-2952(79)90456-8.

DOI:10.1016/0006-2952(79)90456-8

PMID:444312

Abstract

摘要

相似文献

Functional evidence for a second binding site of nicotinic antagonists using phencyclidine derivatives.

Biochem Pharmacol. 1979 Apr 15;28(8):1447-50. doi: 10.1016/0006-2952(79)90456-8.

Sites of action of phencyclidine. II. Interaction with the ionic channel of the nicotinic receptor.苯环己哌啶的作用位点。II. 与烟碱型受体离子通道的相互作用。

Mol Pharmacol. 1980 Sep;18(2):167-78.

Interaction of MK-801 with the nicotinic acetylcholine receptor-associated ion channel from electroplax.MK-801与电鳐的烟碱型乙酰胆碱受体相关离子通道的相互作用。

Eur J Pharmacol. 1989 May 19;164(2):397-8. doi: 10.1016/0014-2999(89)90487-1.

Site of action of phencyclidine. IV. Interaction of phencyclidine and its analogues on ionic channels of the electrically excitable membrane and nicotinic receptor: implications for behavioral effects.

Mol Pharmacol. 1982 May;21(3):637-47.

[3H]Phencyclidine interactions with the nicotinic acetylcholine receptor channel and its inhibition by psychotropic, antipsychotic, opiate, antidepressant, antibiotic, antiviral, and antiarrhythmic drugs.

Mol Pharmacol. 1982 Jul;22(1):72-81.

Effects of thiol modification and Ca++ on agonist-specific state transitions of nicotinic acetylcholine receptor from Torpedo californica electroplax.巯基修饰和钙离子对加州电鳐电板烟碱型乙酰胆碱受体激动剂特异性状态转变的影响。

Life Sci. 1979 May 14;24(20):1893-9. doi: 10.1016/0024-3205(79)90241-8.

Specific binding of [3H]phencyclidines to membrane preparation. Possible interaction with the cholinergic ionophore.

FEBS Lett. 1980 Jan 1;109(1):125-8. doi: 10.1016/0014-5793(80)81325-1.

[3H]Phencyclidine: a probe for the ionic channel of the nicotinic receptor.[3H]苯环己哌啶：一种用于烟碱型受体离子通道的探针。

Proc Natl Acad Sci U S A. 1980 Dec;77(12):7458-62. doi: 10.1073/pnas.77.12.7458.

Amantadine: neuromuscular blockade by suppression of ionic conductance of the acetylcholine receptor.金刚烷胺：通过抑制乙酰胆碱受体的离子电导实现神经肌肉阻滞。

Science. 1978 Feb 17;199(4330):788-90. doi: 10.1126/science.622570.

Binding of perhydrohistrionicotoxin to intact and detergent-solubilized membranes enriched in nicotinic acetylcholine receptor.全氢组胺毒素与富含烟碱型乙酰胆碱受体的完整膜和去污剂增溶膜的结合。

Biochemistry. 1979 May 15;18(10):1868-74. doi: 10.1021/bi00577a004.

引用本文的文献

Ultraviolet light-induced labeling by noncompetitive blockers of the acetylcholine receptor from Torpedo marmorata.用非竞争性阻滞剂对斑纹电鳐乙酰胆碱受体进行紫外线诱导标记。

Proc Natl Acad Sci U S A. 1981 Jun;78(6):3925-9. doi: 10.1073/pnas.78.6.3925.

Phencyclidine interactions with the ionic channel of the acetylcholine receptor and electrogenic membrane.苯环利定与乙酰胆碱受体离子通道及生电膜的相互作用。

Proc Natl Acad Sci U S A. 1980 Feb;77(2):1224-8. doi: 10.1073/pnas.77.2.1224.

Neuropharmacological studies of phencyclidine (PCP)-induced behavioral stimulation in mice.苯环利定（PCP）诱导小鼠行为兴奋的神经药理学研究。

Psychopharmacology (Berl). 1980;71(3):291-7. doi: 10.1007/BF00433064.

Demonstration and affinity labeling of a stereoselective binding site for a benzomorphan opiate on acetylcholine receptor-rich membranes from Torpedo electroplaque.

Proc Natl Acad Sci U S A. 1985 Feb;82(3):940-4. doi: 10.1073/pnas.82.3.940.

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