脑γ-氨基丁酸/苯二氮䓬受体复合物的部分激动剂。 - Suppr

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超能文献

Partial agonists for brain GABA/benzodiazepine receptor complex.

作者信息

Braestrup C, Nielsen M, Krogsgaard-Larsen P, Falch E

出版信息

Nature. 1979 Jul 26;280(5720):331-3. doi: 10.1038/280331a0.

DOI:10.1038/280331a0

PMID:460407

Abstract

摘要

相似文献

Partial agonists for brain GABA/benzodiazepine receptor complex.脑γ-氨基丁酸/苯二氮䓬受体复合物的部分激动剂。

Nature. 1979 Jul 26;280(5720):331-3. doi: 10.1038/280331a0.

Influence of GABA receptor agonists and antagonists on the binding of 3H-diazepam to the benzodiazepine receptor.

Eur J Pharmacol. 1978 Nov 1;52(1):129-32. doi: 10.1016/0014-2999(78)90031-6.

Two or more conformations of benzodiazepine receptors depending on GABA receptors and other variables.苯二氮䓬受体的两种或更多种构象取决于γ-氨基丁酸（GABA）受体及其他变量。

Adv Biochem Psychopharmacol. 1980;21:301-12.

Stimulation of benzodiazepine receptor binding by gamma-aminobutyric acid.γ-氨基丁酸对苯二氮䓬受体结合的刺激作用。

Proc Natl Acad Sci U S A. 1979 Feb;76(2):1004-6. doi: 10.1073/pnas.76.2.1004.

Modulation of [3H]diazepam binding in rat cortical membranes by GABAA agonists.γ-氨基丁酸A受体激动剂对大鼠皮层膜中[3H]地西泮结合的调节作用

J Neurochem. 1985 Apr;44(4):1162-7. doi: 10.1111/j.1471-4159.1985.tb08739.x.

GABA reduces binding of 3H-methyl beta-carboline-3-carboxylate to brain benzodiazepine receptors.γ-氨基丁酸可降低³H-甲基β-咔啉-3-羧酸与脑苯二氮䓬受体的结合。

Nature. 1981 Dec 3;294(5840):472-4. doi: 10.1038/294472a0.

THIP and isoguvacine are partial agonists of GABA-stimulated benzodiazepine receptor binding.THIP和异谷氨酰胺是γ-氨基丁酸（GABA）刺激的苯二氮䓬受体结合的部分激动剂。

Eur J Pharmacol. 1979 Oct 15;58(4):485-8. doi: 10.1016/0014-2999(79)90321-2.

The inhibition of GABA-stimulated benzodiazepine binding by a convulsant benzodiazepine.一种惊厥性苯二氮䓬对γ-氨基丁酸刺激的苯二氮䓬结合的抑制作用。

Life Sci. 1980 Apr 28;26(17):1441-5. doi: 10.1016/0024-3205(80)90047-8.

The GABA agonist THIP a muscimol analogue, does not interfere with the benzodiazepine binding site on rats cortical membranes.GABA 激动剂 THIP（一种蝇蕈醇类似物）不干扰大鼠皮质膜上的苯二氮䓬结合位点。

Neurosci Lett. 1979 Apr;12(1):65-8. doi: 10.1016/0304-3940(79)91481-2.

The insensitivity of developing benzodiazepine receptors to chronic treatment with diazepam, GABA and muscimol in brain cell cultures.

Brain Res. 1981 Apr 6;210(1-2):471-4. doi: 10.1016/0006-8993(81)90929-x.

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Cortical GABAergic Dysfunction in Stress and Depression: New Insights for Therapeutic Interventions.应激与抑郁中的皮质GABA能功能障碍：治疗干预的新见解

Front Cell Neurosci. 2019 Mar 12;13:87. doi: 10.3389/fncel.2019.00087. eCollection 2019.

GABA receptor: Positive and negative allosteric modulators.GABA 受体：正变构调节剂和负变构调节剂。

Neuropharmacology. 2018 Jul 1;136(Pt A):10-22. doi: 10.1016/j.neuropharm.2018.01.036. Epub 2018 Jan 31.

Analysis of γ-aminobutyric acid (GABA) type A receptor subtypes using isosteric and allosteric ligands.使用等排体和变构配体分析γ-氨基丁酸（GABA）A型受体亚型

Neurochem Res. 2014 Oct;39(10):1924-41. doi: 10.1007/s11064-014-1382-3. Epub 2014 Jul 12.

Characteristics of GABAB receptor binding sites on rat whole brain synaptic membranes. 1983.大鼠全脑突触膜上GABAB受体结合位点的特征。1983年。

Br J Pharmacol. 1997 Feb;120(4 Suppl):452-67; discussion 450-1. doi: 10.1111/j.1476-5381.1997.tb06835.x.

Interaction among alfaxalone, pregnenolone sulfate, and two GABAA agonists on hippocampal slices.阿法沙龙、硫酸孕烯醇酮和两种GABAA激动剂在海马切片上的相互作用。

Cell Mol Neurobiol. 1996 Jun;16(3):427-31. doi: 10.1007/BF02088108.

L-lysine is a barbiturate-like anticonvulsant and modulator of the benzodiazepine receptor.L-赖氨酸是一种巴比妥酸盐样抗惊厥药和苯二氮䓬受体调节剂。

Neurochem Res. 1995 Aug;20(8):931-7. doi: 10.1007/BF00970739.

Nigral actions of GABA agonists are enhanced by chronic fluphenazine and differentiated by concomitant flurazepam.慢性氟奋乃静可增强GABA激动剂的黑质作用，且与同时使用氟西泮的作用有所区别。

Psychopharmacology (Berl). 1982;76(3):294-8. doi: 10.1007/BF00432565.

Methylphenidate, apomorphine, THIP, and diazepam in monkeys: dopamine-GABA behavior related to psychoses and tardive dyskinesia.猴子体内的哌甲酯、阿扑吗啡、THIP和地西泮：与精神病和迟发性运动障碍相关的多巴胺-γ-氨基丁酸行为

Psychopharmacology (Berl). 1984;82(1-2):131-4. doi: 10.1007/BF00426396.

Binding of 3H-DMCM to benzodiazepine receptors; chloride dependent allosteric regulation mechanisms.3H-DMCM与苯二氮䓬受体的结合；氯离子依赖性变构调节机制。

J Neural Transm. 1983;58(1-2):83-98. doi: 10.1007/BF01249127.

Characteristics of GABAB receptor binding sites on rat whole brain synaptic membranes.大鼠全脑突触膜上GABAB受体结合位点的特征

Br J Pharmacol. 1983 Jan;78(1):191-206. doi: 10.1111/j.1476-5381.1983.tb09380.x.

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