硫脲类化合物对碘甲状腺原氨酸5'-脱碘酶的抑制作用；构效关系 - Suppr

Suppr

超能文献

Inhibition of iodothyronine 5'-deiodinase by thioureylenes; structure--activity relationship.

作者信息

Visser T J, van Overmeeren E, Fekkes D, Docter R, Hennemann G

出版信息

FEBS Lett. 1979 Jul 15;103(2):314-8. doi: 10.1016/0014-5793(79)81352-6.

DOI:10.1016/0014-5793(79)81352-6

PMID:467676

Abstract

摘要

相似文献

Inhibition of iodothyronine 5'-deiodinase by thioureylenes; structure--activity relationship.硫脲类化合物对碘甲状腺原氨酸5'-脱碘酶的抑制作用；构效关系

FEBS Lett. 1979 Jul 15;103(2):314-8. doi: 10.1016/0014-5793(79)81352-6.

Inhibition of iodothyronine deiodinase by phenolphthalein dyes: structure--activity relationship.酚酞染料对碘甲状腺原氨酸脱碘酶的抑制作用：构效关系

FEBS Lett. 1982 Jan 11;137(1):40-4. doi: 10.1016/0014-5793(82)80310-4.

Mechanism of inhibition of iodothyronine-5'-deiodinase by thioureylenes and sulfite.硫脲类和亚硫酸盐对碘甲状腺原氨酸-5'-脱碘酶的抑制机制。

Biochim Biophys Acta. 1980 Feb 14;611(2):371-8. doi: 10.1016/0005-2744(80)90074-1.

Inactivation and affinity-labeling of rat liver iodothyronine deiodinase with N-bromoacetyl-3,3',5-triiodothyronine.用N-溴乙酰基-3,3',5-三碘甲状腺原氨酸对大鼠肝脏碘甲状腺原氨酸脱碘酶进行失活和亲和标记

Biochem Biophys Res Commun. 1984 Oct 30;124(2):475-83. doi: 10.1016/0006-291x(84)91578-x.

Modification of rat liver iodothyronine 5'-deiodinase activity with diethylpyrocarbonate and rose bengal; evidence for an active site histidine residue.

Biochem Biophys Res Commun. 1984 Apr 16;120(1):28-36. doi: 10.1016/0006-291x(84)91409-8.

Thiourea and cyanamide as inhibitors of thyroid peroxidase: the role of iodide.硫脲和氰胺作为甲状腺过氧化物酶的抑制剂：碘化物的作用。

Endocrinology. 1979 Apr;104(4):919-24. doi: 10.1210/endo-104-4-919.

Substrate requirement for inactivation of iodothyronine-5'-deiodinase activity by thiouracil.硫脲使碘甲状腺原氨酸5'-脱碘酶失活的底物需求。

Biochim Biophys Acta. 1981 Apr 14;658(2):202-8. doi: 10.1016/0005-2744(81)90290-4.

Antihormonal effects of plant extracts: iodothyronine deiodinase of rat liver is inhibited by extracts and secondary metabolites of plants.

Horm Metab Res. 1984 Apr;16(4):188-92. doi: 10.1055/s-2007-1014739.

Inhibition of rat liver iodothyronine deiodinase. Interaction of aurones with the iodothyronine ligand-binding site.大鼠肝脏碘甲状腺原氨酸脱碘酶的抑制作用。奥酮与碘甲状腺原氨酸配体结合位点的相互作用。

J Biol Chem. 1986 Sep 5;261(25):11623-30.

5'-Iodothyronine deiodinase of rat liver: activity in microsomes prepared by various methods, solubilization by detergents and partial purification.

Biochim Biophys Acta. 1985 Aug 16;841(2):173-85. doi: 10.1016/0304-4165(85)90019-4.

引用本文的文献

An AOP-based alternative testing strategy to predict the impact of thyroid hormone disruption on swim bladder inflation in zebrafish.一种基于 AOP 的替代测试策略，用于预测甲状腺激素干扰对斑马鱼鳔充气的影响。

Aquat Toxicol. 2018 Jul;200:1-12. doi: 10.1016/j.aquatox.2018.04.009. Epub 2018 Apr 21.

Se- and s-based thiouracil and methimazole analogues exert different inhibitory mechanisms on type 1 and type 2 deiodinases.硒代和硫代尿嘧啶和甲巯咪唑类似物对 1 型和 2 型脱碘酶发挥不同的抑制机制。

Eur Thyroid J. 2013 Dec;2(4):252-8. doi: 10.1159/000355288. Epub 2013 Nov 27.

Identification of thyroid hormone receptor active compounds using a quantitative high-throughput screening platform.使用定量高通量筛选平台鉴定甲状腺激素受体活性化合物。

Curr Chem Genom Transl Med. 2014 Mar 7;8:36-46. doi: 10.2174/2213988501408010036. eCollection 2014.

Thyroid-disrupting chemicals: interpreting upstream biomarkers of adverse outcomes.甲状腺干扰化学物质：解读不良后果的上游生物标志物。

Environ Health Perspect. 2009 Jul;117(7):1033-41. doi: 10.1289/ehp.0800247. Epub 2009 Feb 12.

Bioinorganic chemistry in thyroid gland: effect of antithyroid drugs on peroxidase-catalyzed oxidation and iodination reactions.甲状腺中的生物无机化学：抗甲状腺药物对过氧化物酶催化的氧化和碘化反应的影响。

Bioinorg Chem Appl. 2006;2006:23214. doi: 10.1155/BCA/2006/23214. Epub 2006 Nov 12.

Structural requirements of thiol compounds in the inhibition of human liver iodothyronine 5'-deiodinase.硫醇化合物对人肝脏碘甲状腺原氨酸5'-脱碘酶抑制作用的结构要求

Biochem J. 1984 Jan 15;217(2):485-91. doi: 10.1042/bj2170485.

文献AI研究员

20分钟写一篇综述，助力文献阅读效率提升50倍。

立即体验

用中文搜PubMed

大模型驱动的PubMed中文搜索引擎

马上搜索

文档翻译

学术文献翻译模型，支持多种主流文档格式。

立即体验