Conformation of histamine derivatives. 3. A relationship between conformation and pharmacological activity.
作者信息
Ganellin C R
出版信息
J Med Chem. 1973 Jun;16(6):620-3. doi: 10.1021/jm00264a009.
PMID:4714992
Abstract
摘要
相似文献
1
Conformation of histamine derivatives. 3. A relationship between conformation and pharmacological activity.组胺衍生物的构象。3. 构象与药理活性之间的关系。
J Med Chem. 1973 Jun;16(6):620-3. doi: 10.1021/jm00264a009.
2
Proceedings: Structure-action-relationships of histamine analogues.论文集：组胺类似物的构效关系
Naunyn Schmiedebergs Arch Pharmacol. 1974;282(Suppl):suppl 282:R90.
3
Stable conformations of histamine by empirical method.通过经验方法得到的组胺稳定构象。
J Theor Biol. 1975 Sep;53(2):333-40. doi: 10.1016/s0022-5193(75)80008-7.
4
Conformation of histamine derivatives. 2. Molecular orbital calculations of preferred conformations in relation to dual receptor activity.组胺衍生物的构象。2. 与双重受体活性相关的优选构象的分子轨道计算。
J Med Chem. 1973 Jun;16(6):616-20. doi: 10.1021/jm00264a008.
5
Conformationally restricted analogs of histamine H1 receptor antagonists. Trans- and cis-1,5-Diphenyl-3-dimethylaminopyrrolidine.
J Med Chem. 1973 Sep;16(9):963-8. doi: 10.1021/jm00267a001.
6
Conformationally restricted analogs of histamine H1 receptor antagonists: trans and cis-1-benzyl-3-dimethylamino-6-phenylpiperidine.组胺H1受体拮抗剂的构象受限类似物：反式和顺式-1-苄基-3-二甲基氨基-6-苯基哌啶
J Med Chem. 1976 Jan;19(1):117-22. doi: 10.1021/jm00223a020.
7
Tautomerism and the receptor action of histamine: a mechanistic model.组胺的互变异构与受体作用：一种机制模型
Mol Pharmacol. 1976 Sep;12(5):738-45.
8
Conformation of histamine derivatives. 5. Molecular orbital calculation of the H1-receptor "essential" conformation of histamine.组胺衍生物的构象。5. 组胺H1受体“基本”构象的分子轨道计算。
J Med Chem. 1975 Jul;18(7):662-6. doi: 10.1021/jm00241a003.
9
[Burimamid and metiamid, a new pharmacological principle].[布立马胺和甲硫米特，一种新的药理学原理]
Internist (Berl). 1974 Mar;15(3):177-8.
10
[Effects of histamine and its derivatives on the excitability of a giant identifiable neuron of Achatina fulica Férussac. A histaminergic receptor different from H1 and H2].
C R Seances Soc Biol Fil. 1976;170(5):1118-26.
引用本文的文献
1
Classification and biological distribution of histamine receptor sub-types. 1975.组胺受体亚型的分类及生物学分布。1975年。
Agents Actions. 1994 Dec;43(3-4):97-115; discussion 116. doi: 10.1007/BF01986677.
2
Dimaprit, [S-[3-(N,N-dimethylamino)propyl]isothiourea]. A highly specific histamine H2-receptor agonist. Part 2. Structure-activity considerations. 1977.二甲双胍，[S-[3-(N,N-二甲基氨基)丙基]异硫脲]。一种高度特异性的组胺H2受体激动剂。第2部分。构效关系探讨。1977年。
Agents Actions. 1994 Dec;43(3-4):139-43. doi: 10.1007/BF01986680.
3
Histamine receptor activation by unsaturated (allyl and propargyl) homologs of histamine.组胺的不饱和（烯丙基和炔丙基）同系物对组胺受体的激活作用。
Agents Actions. 1985 Dec;17(2):138-44. doi: 10.1007/BF01966582.
4
The effects of L-histidine and of specific histamine receptor agonists, on the expression of morphine tolerance and physical dependence in mice.L-组氨酸及特定组胺受体激动剂对小鼠吗啡耐受性和身体依赖性表达的影响。
Agents Actions. 1976 Sep;6(5):569-76. doi: 10.1007/BF01971571.
5
Dimaprit, (S-[3-(N,N-dimethylamino)propyl]isothiourea). A highly specific histamine H2-receptor agonist. Part 2. Structure-activity considerations.地马普明，（S-[3-(N,N-二甲基氨基)丙基]异硫脲）。一种高度特异性的组胺H2受体激动剂。第2部分。构效关系探讨。
Agents Actions. 1977 Mar;7(1):39-43. doi: 10.1007/BF01964879.
6
Tautomerism of 4-methylhistamine--effect of the methyl substituent [proceedings].4-甲基组胺的互变异构——甲基取代基的影响[会议论文集]
Agents Actions. 1979 Apr;9(1):27-8. doi: 10.1007/BF02024092.
7
Relative conformational rigidity in oxytocin and (1-penicillamine)-oxytocin: a proposal for the relationship of conformational flexibility to peptide hormone agonism and antagonism.催产素和（1-青霉胺）-催产素中的相对构象刚性：关于构象灵活性与肽类激素激动作用和拮抗作用关系的一项提议。
Proc Natl Acad Sci U S A. 1977 Apr;74(4):1373-7. doi: 10.1073/pnas.74.4.1373.
8
Histamine and its metabolism in mammals. Part II: Catabolism of histamine and histamine liberation.组胺及其在哺乳动物体内的代谢。第二部分：组胺的分解代谢与组胺释放
Agents Actions. 1975 Aug;5(3):183-225. doi: 10.1007/BF02026434.
9
Classification and biological distribution of histamine receptor sub-types.组胺受体亚型的分类及生物学分布
Agents Actions. 1975 Oct;5(4):277-95. doi: 10.1007/BF02205232.
Zotero 插件